SCHEMBL6565445

SCHEMBL6565445

CCOC(=O)CN(C(=O)Nc1cc(C(F)(F)F)c(C#CCNc2ccc(C(=N)N)cc2)cc1C(F)(F)F)C(C)C

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.36
ITGA2B P08514 2/20 0.36
F7 P08709 3/20 0.34
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
PAX8 Q06710 1/20 0.33
F2 P00734 8/20 0.32
PLAU P00749 6/20 0.32
HPN P05981 4/20 0.32
F10 P00742 6/20 0.31
PRSS1 P07477 3/20 0.31
KLK1 P06870 1/20 0.30
PLAT P00750 1/20 0.30
PRSS2 P07478 1/20 0.30
F3 P13726 1/20 0.30
PRSS3 P35030 1/20 0.30
NQO2 P16083 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563559 0.95 ITGB3 (0.36) ITGB3ITGA2BF7NPC1ALDH1A1
SCHEMBL6565368 0.91 ITGB3 (0.37) ITGB3ITGA2BF7HTTF2
SCHEMBL6563598 0.90 F7 (0.38) ITGB3ITGA2BF7NPC1ALDH1A1
SCHEMBL6563746 0.85 F7 (0.37) ITGB3ITGA2BF7NPC1ALDH1A1
SCHEMBL7670894 0.85 ITGB3 (0.39) ITGB3ITGA2BF7F2PLAU
SCHEMBL6565399 0.84 ITGB3 (0.37) ITGB3ITGA2BF7F2PLAU
SCHEMBL6561894 0.83 ITGB3 (0.40) ITGB3ITGA2BF7NPC1RAB9A
SCHEMBL6563523 0.83 ITGB3 (0.37) ITGB3ITGA2BF7RAB9AF2
SCHEMBL6563366 0.82 ITGB3 (0.39) ITGB3ITGA2BF7ALDH1A1F2
SCHEMBL6565440 0.81 F7 (0.36) ITGB3ITGA2BF7NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed