SCHEMBL6563695

SCHEMBL6563695

CCc1cc(CC)n(-c2ccc(C#CCNc3ccc(C(=N)NC(=O)OC(C)(C)C)cc3)cc2C)n1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.34
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565301 0.90 CA12 (0.31) CA12CA1CA2CA9
SCHEMBL6563913 0.82 CA12 (0.33) CA12CA1CA2CA9
SCHEMBL6561879 0.77 PTPN11 (0.38) PTPN11
SCHEMBL6565533 0.76 ACACB (0.45) PTPN11
SCHEMBL6563526 0.75 PTPN11 (0.38) PTPN11
SCHEMBL6561973 0.74 JAK1 (0.38) PTPN11
SCHEMBL6565215 0.73 PIK3CA (0.38) PTPN11
SCHEMBL6563355 0.72 PTPN11 (0.47) PTPN11CA12CA1CA2
SCHEMBL6563070 0.72 PTPN11 (0.44) PTPN11
SCHEMBL6565417 0.72 PTPN11 (0.36) PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed