SCHEMBL6563913

SCHEMBL6563913

CCc1cc(CC)n(-c2ccc(C#CCNc3ccc(C(=N)N)cc3)cc2C)n1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
PRSS1 P07477 9/20 0.33
F2 P00734 3/20 0.32
PRSS2 P07478 2/20 0.32
PRSS3 P35030 2/20 0.32
TMPRSS6 Q8IU80 2/20 0.32
ST14 Q9Y5Y6 2/20 0.32
F7 P08709 2/20 0.32
F10 P00742 1/20 0.32
KLK1 P06870 1/20 0.31
KLK5 Q9Y337 1/20 0.31
EGLN1 Q9GZT9 1/20 0.31
F3 P13726 1/20 0.31
ITGB3 P05106 1/20 0.30
ITGA2B P08514 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6564407 0.88 CA12 (0.34) CA12CA1CA2CA9PRSS1
SCHEMBL6563695 0.82 PTPN11 (0.34) CA12CA1CA2CA9
SCHEMBL6771187 0.79 MAPT (0.38) CA12CA1CA2CA9PRSS1
SCHEMBL6563544 0.76 RXRA (0.38) PRSS1F2PRSS2PRSS3F10
SCHEMBL6563546 0.75 F10 (0.38) F2F7F10F3ITGB3
SCHEMBL6562124 0.75 KLK5 (0.47) PRSS1F2KLK1KLK5
SCHEMBL6565301 0.71 CA12 (0.31) CA12CA1CA2CA9
SCHEMBL7675036 0.71 F10 (0.42) CA1CA2PRSS1F2PRSS2
SCHEMBL6563461 0.71 PRSS1 (0.49) PRSS1F2PRSS2PRSS3TMPRSS6
SCHEMBL6565349 0.70 F2 (0.38) PRSS1F2PRSS2PRSS3TMPRSS6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed