SCHEMBL6563070

SCHEMBL6563070

CC(C)(C)OC(=O)NC(=N)c1ccc(NCC#Cc2ccc(C(=O)c3ccncc3)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.44
CYP17A1 P05093 4/20 0.43
KMT2A Q03164 3/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35
ADRB3 P13945 1/20 0.35
PPARG P37231 6/20 0.35
PPARA Q07869 6/20 0.35
PPARD Q03181 2/20 0.35
NAMPT P43490 1/20 0.35
MEN1 O00255 2/20 0.34
RAB9A P51151 1/20 0.34
NR1H4 Q96RI1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563676 0.90 NAMPT (0.42) PTPN11CYP17A1KMT2APPARGPPARA
SCHEMBL6563283 0.84 PTPN11 (0.46) PTPN11CYP17A1NR1H4
SCHEMBL6565434 0.83 PTPN11 (0.41) PTPN11KMT2AADRB2ADRB1ADRB3
SCHEMBL7686729 0.82 PTPN11 (0.43) PTPN11KMT2ANAMPTMEN1
SCHEMBL7674981 0.82 ABL1 (0.43) PTPN11KMT2ANAMPTMEN1RAB9A
SCHEMBL6563355 0.82 PTPN11 (0.47) PTPN11CYP17A1PPARGPPARAPPARD
SCHEMBL6565384 0.81 GRM5 (0.46) PTPN11KMT2ANAMPTMEN1
SCHEMBL6561813 0.80 PTPN11 (0.42) PTPN11NAMPT
SCHEMBL7677130 0.80 PRSS1 (0.41) KMT2ANPSR1MEN1
SCHEMBL6561858 0.79 GRM5 (0.47) PTPN11KMT2ANAMPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed