SCHEMBL6562124

SCHEMBL6562124

Cc1cc(C#CCNc2ccc(C(=N)N)cc2)ccc1-n1c(C)nc2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 4/20 0.47
KLK1 P06870 3/20 0.47
TSHR P16473 1/20 0.42
F2 P00734 6/20 0.34
HPGD P15428 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
BMI1 P35226 1/20 0.34
ASIC3 Q9UHC3 1/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33
TUBB4B P68371 1/20 0.33
TUBB3 Q13509 1/20 0.33
TUBB2A Q13885 1/20 0.33
TUBB8 Q3ZCM7 1/20 0.33
TUBA3E Q6PEY2 1/20 0.33
TUBA1A Q71U36 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6562437 0.80 KLK5 (0.47) KLK5KLK1TSHRHTTTP53
SCHEMBL6563913 0.75 CA12 (0.33) KLK5KLK1F2PRSS1
SCHEMBL6563277 0.72 F2 (0.41) KLK5KLK1F2ASIC3PLG
SCHEMBL7071377 0.71 KLK5 (0.41) KLK5KLK1TSHRF2HPGD
Hydrochloric Acid SCHEMBL6943397 0.71 KLK5 (0.41) KLK5KLK1TSHRF2HPGD
SCHEMBL6563255 0.71 PRSS1 (0.44) KLK5KLK1F2ASIC3PLG
SCHEMBL6563544 0.70 RXRA (0.38) F2HPGDPRSS1ALDH1A1CYP2C19
SCHEMBL6563461 0.70 PRSS1 (0.49) KLK5KLK1F2PLGPRSS1
SCHEMBL7675036 0.68 F10 (0.42) KLK5KLK1F2PLGPRSS1
SCHEMBL6561958 0.68 ACACB (0.49) KLK5KLK1F2HPGDPLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed