SCHEMBL6565221

SCHEMBL6565221

Cc1cc(C(=O)N2CCOCC2)ccc1C#CCNc1ccc(C(=N)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.41
HPGD P15428 3/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HSP90AA1 P07900 2/20 0.38
HSP90AB1 P08238 2/20 0.38
B3GNT2 Q9NY97 1/20 0.38
CD274 Q9NZQ7 1/20 0.37
GAA P10253 2/20 0.37
RAB9A P51151 2/20 0.36
BTK Q06187 1/20 0.36
KMT2A Q03164 2/20 0.36
NPC1 O15118 1/20 0.36
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.35
F10 P00742 1/20 0.35
NAMPT P43490 1/20 0.35
GLA P06280 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563568 0.92 CNR2 (0.39) HPGDGAAKMT2APOLBNAMPT
SCHEMBL6561973 0.86 JAK1 (0.38) SMN1; SMN2HPGDCD274KMT2A
SCHEMBL6563686 0.83 F10 (0.46) SMN1; SMN2HPGDKDM4EALDH1A1GAA
SCHEMBL6561938 0.83 ABL1 (0.36) HPGDALDH1A1GAARAB9AKMT2A
SCHEMBL6563605 0.83 GAA (0.37) HPGDALDH1A1GAAKMT2ANPC1
SCHEMBL7686729 0.79 PTPN11 (0.43) SMN1; SMN2HPGDKDM4EALDH1A1KMT2A
SCHEMBL7674981 0.79 ABL1 (0.43) SMN1; SMN2HPGDKDM4EALDH1A1GAA
SCHEMBL6563229 0.78 PLAU (0.37) KDM4EALDH1A1RAB9AKMT2ANPC1
SCHEMBL6565533 0.78 ACACB (0.45) ALDH1A1GAARAB9AKMT2AF10
SCHEMBL6563627 0.77 PTPN11 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed