SCHEMBL6563605

SCHEMBL6563605

Cc1cc(C(=O)N2CCCC2C)ccc1C#CCNc1ccc(C(=N)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 2/20 0.36
NAMPT P43490 2/20 0.36
HTT P42858 1/20 0.36
HRH3 Q9Y5N1 3/20 0.36
MEN1 O00255 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
PDK2 Q15119 1/20 0.35
NPC1 O15118 1/20 0.34
HSD11B1 P28845 1/20 0.34
MAP4K1 Q92918 1/20 0.33
AVPR2 P30518 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563752 0.91 GAA (0.35) GAAALDH1A1HPGDNAMPTHTT
SCHEMBL6563591 0.91 LRRK2 (0.39) GAAALDH1A1HPGDNAMPTHTT
SCHEMBL6563002 0.88 HRH3 (0.42) GAAALDH1A1HPGDNAMPTHRH3
SCHEMBL6565417 0.87 PTPN11 (0.36) GAAALDH1A1HPGDNAMPTHRH3
SCHEMBL6563568 0.87 CNR2 (0.39) GAAHPGDNAMPTHTTMEN1
SCHEMBL6563507 0.85 KCNK3 (0.31) GAAALDH1A1HPGDNAMPTHTT
SCHEMBL6565356 0.84 GAA (0.42) GAAALDH1A1HPGDNAMPTHTT
SCHEMBL6565221 0.83 SMN1; SMN2 (0.41) GAAALDH1A1HPGDNAMPTMAPK1
SCHEMBL6561835 0.82 PTPN11 (0.35) GAAALDH1A1HPGDNAMPTHTT
SCHEMBL6561938 0.79 ABL1 (0.36) GAAALDH1A1HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed