SCHEMBL6565356

SCHEMBL6565356

Cc1cc(C(=O)N2CCCC2C)ccc1C#CCNc1ccc(C(=N)N)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 2/20 0.42
NAMPT P43490 2/20 0.41
MEN1 O00255 1/20 0.39
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.39
HTT P42858 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
HSD11B1 P28845 1/20 0.38
F2 P00734 2/20 0.37
MAP4K1 Q92918 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
PDK2 Q15119 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563410 0.90 GAA (0.40) GAAALDH1A1HPGDNAMPTMEN1
SCHEMBL6563266 0.88 LRRK2 (0.42) GAAALDH1A1HPGDNAMPTMEN1
SCHEMBL6561970 0.85 GAA (0.49) GAAALDH1A1HPGDNAMPTCA12
SCHEMBL6565512 0.85 GAA (0.40) GAAALDH1A1HPGDNAMPTMEN1
SCHEMBL6564299 0.85 GAA (0.36) GAAALDH1A1HPGDNAMPTMEN1
SCHEMBL7671074 0.84 F10 (0.43) GAAALDH1A1HPGDMEN1KMT2A
SCHEMBL6563605 0.84 GAA (0.37) GAAALDH1A1HPGDNAMPTMEN1
SCHEMBL6561673 0.82 PRSS1 (0.35) GAAALDH1A1HPGDNAMPTMEN1
SCHEMBL6563686 0.80 F10 (0.46) GAAALDH1A1HPGDNAMPTKMT2A
SCHEMBL6563261 0.79 HSD11B1 (0.38) GAAALDH1A1HPGDNAMPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed