SCHEMBL6563266

SCHEMBL6563266

COc1cc(C(=O)N2CCCC2C)ccc1C#CCNc1ccc(C(=N)N)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.42
HSD11B1 P28845 4/20 0.41
GAA P10253 2/20 0.40
HPGD P15428 1/20 0.40
NAMPT P43490 1/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
ROCK2 O75116 2/20 0.37
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
HTT P42858 1/20 0.37
HRH3 Q9Y5N1 2/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565356 0.88 GAA (0.42) HSD11B1GAAHPGDNAMPTALDH1A1
SCHEMBL6563591 0.85 LRRK2 (0.39) LRRK2HSD11B1GAAHPGDNAMPT
SCHEMBL6561970 0.83 GAA (0.49) HSD11B1GAAHPGDNAMPTALDH1A1
SCHEMBL6563410 0.82 GAA (0.40) HSD11B1GAAHPGDNAMPTALDH1A1
SCHEMBL6565512 0.81 GAA (0.40) HSD11B1GAAHPGDNAMPTALDH1A1
SCHEMBL6563261 0.78 HSD11B1 (0.38) HSD11B1GAAHPGDNAMPTALDH1A1
SCHEMBL6563696 0.78 HPGD (0.37) LRRK2HSD11B1GAAHPGDNAMPT
SCHEMBL6564299 0.77 GAA (0.36) HSD11B1GAAHPGDNAMPTALDH1A1
SCHEMBL6561673 0.77 PRSS1 (0.35) HSD11B1GAAHPGDNAMPTALDH1A1
SCHEMBL6566003 0.77 F2 (0.37) HSD11B1GAAHPGDNAMPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed