SCHEMBL6565633

SCHEMBL6565633

O=C(Cc1cc(Cl)c(O)c(Cl)c1)NC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
TDP1 Q9NUW8 2/20 0.49
EPHX2 P34913 1/20 0.47
ALDH1A1 P00352 4/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
KDM4E B2RXH2 1/20 0.46
HPGD P15428 1/20 0.46
RAB9A P51151 2/20 0.46
NPC1 O15118 1/20 0.46
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
CNR2 P34972 1/20 0.43
JAK2 O60674 1/20 0.43
LMNA P02545 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10922194 0.78 HTT (0.76) HTTNPSR1TDP1EPHX2ALDH1A1
SCHEMBL19798449 0.76 KMT2A (0.72) HTTEPHX2ALDH1A1MEN1KMT2A
SCHEMBL4348906 0.75 EPHX2 (0.73) HTTNPSR1EPHX2MEN1KMT2A
SCHEMBL19798759 0.74 ALDH1A1 (0.68) HTTEPHX2ALDH1A1MEN1KMT2A
SCHEMBL8848470 0.71 CNR2 (0.56) HTTNPSR1EPHX2ALDH1A1KDM4E
SCHEMBL13596196 0.70 NPC1 (0.54) EPHX2ALDH1A1MEN1KMT2ARAB9A
SCHEMBL6567675 0.70 P2RX7 (0.65) NPSR1EPHX2MEN1KMT2APOLB
SCHEMBL13596178 0.69 ADRB2 (0.59) EPHX2ALDH1A1MEN1KMT2ARAB9A
SCHEMBL4346873 0.69 EPHX2 (0.57) NPSR1EPHX2MAPT
SCHEMBL9334741 0.69 TSHR (0.61) HTTEPHX2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed