SCHEMBL6565641

SCHEMBL6565641

Cc1ccc(NC(=O)Nc2ccc(C#N)cc2)c(O)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 3/20 0.68
CXCR1 P25024 2/20 0.67
MAPT P10636 5/20 0.54
LMNA P02545 3/20 0.54
TSHR P16473 1/20 0.54
HTT P42858 1/20 0.54
NLRP3 Q96P20 1/20 0.54
MEN1 O00255 5/20 0.54
KMT2A Q03164 5/20 0.54
ALDH1A1 P00352 4/20 0.54
RAB9A P51151 3/20 0.52
KDM4E B2RXH2 2/20 0.52
MAPK1 P28482 2/20 0.52
SAE1 Q9UBE0 1/20 0.52
UBA2 Q9UBT2 1/20 0.52
POLB P06746 1/20 0.52
PKM P14618 1/20 0.52
IL18 Q14116 1/20 0.52
CA12 O43570 2/20 0.52
CA1 P00915 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4359536 0.86 CXCR1 (0.70) CXCR2CXCR1MAPTLMNATSHR
SCHEMBL11054936 0.83 MAPT (0.69) MAPTLMNATSHRHTTNLRP3
SCHEMBL8982693 0.83 CXCR2 (0.67) CXCR2CXCR1MAPTLMNATSHR
SCHEMBL6567616 0.81 CXCR2 (0.73) CXCR2MAPTLMNAHTTNLRP3
SCHEMBL12376726 0.81 PABPC1 (0.52) CXCR2CXCR1MAPTLMNAMEN1
SCHEMBL5605320 0.81 CXCR2 (1.00) CXCR2CXCR1MAPTTSHRHTT
SCHEMBL10957092 0.81 CXCR2 (0.60) CXCR2CXCR1MAPTLMNATSHR
SCHEMBL5594683 0.80 CXCR1 (0.70) CXCR2CXCR1MAPTLMNATSHR
SCHEMBL7489930 0.80 CXCR2 (1.00) CXCR2CXCR1MAPTLMNATSHR
SCHEMBL9267208 0.79 CXCR1 (0.70) CXCR2CXCR1MAPTLMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed