SCHEMBL6565811

SCHEMBL6565811

CC(CCOC(=O)NCc1ccccc1)CC(=O)NC(C)(C#N)COCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSS P25774 11/20 0.40
CTSL P07711 8/20 0.38
CTSB P07858 3/20 0.38
CTSK P43235 3/20 0.38
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PLAU P00749 1/20 0.36
MCL1 Q07820 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563827 0.79 CTSS (0.47) CTSSCTSLCTSBCTSKCHRNB2
SCHEMBL7438096 0.76 CTSS (0.42) CTSSCTSLCTSBCTSKPLAU
SCHEMBL3895827 0.76 CTSS (0.43) CTSSCTSLCTSBCTSK
SCHEMBL6567353 0.75 CHRNB2 (0.42) CTSSCTSLCTSBCTSKCHRNB2
SCHEMBL6182445 0.73 CTSS (0.49) CTSSCTSLCTSBCTSKLMNA
SCHEMBL6565460 0.73 CHRNB2 (0.41) CTSSCTSLCTSBCTSKCHRNB2
SCHEMBL3893933 0.72 CTSS (0.39) CTSSCTSLCTSBCTSK
SCHEMBL6565044 0.69 CHRNB2 (0.41) CTSSCTSLCTSBCTSKCHRNB2
SCHEMBL6182870 0.68 CTSS (0.53) CTSSCTSLCTSBCTSK
Hydrochloric Acid SCHEMBL28665674 0.67 CHRNB2 (0.50) CHRNB2CHRNB4CHRNA3CHRNA4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed