SCHEMBL6567353

SCHEMBL6567353

CC(CC#N)CCNC(=O)CC(C)CCOC(=O)NCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA4 P43681 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
MCL1 Q07820 1/20 0.41
HPGD P15428 3/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
CTSS P25774 3/20 0.39
CTSL P07711 2/20 0.39
CTSB P07858 1/20 0.39
CTSK P43235 1/20 0.39
ALDH1A1 P00352 3/20 0.38
PLA2G1B P04054 1/20 0.38
ATG4B Q9Y4P1 1/20 0.38
MAPT P10636 1/20 0.38
KCNA5 P22460 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
CASP3 P42574 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563827 0.88 CTSS (0.47) CHRNB2CHRNB4CHRNA3CHRNA4L3MBTL1
SCHEMBL6565460 0.88 CHRNB2 (0.41) CHRNB2CHRNB4CHRNA3CHRNA4L3MBTL1
SCHEMBL6183160 0.86 CTSS (0.49) L3MBTL1CTSSCTSLCTSBCTSK
SCHEMBL6183204 0.78 CTSS (0.49) L3MBTL1CTSSCTSLCTSBCTSK
SCHEMBL7456077 0.77 CTSS (0.57) L3MBTL1CTSSCTSLCTSBCTSK
SCHEMBL6181806 0.77 CTSS (0.57) L3MBTL1CTSSCTSLCTSBCTSK
SCHEMBL6567346 0.77 L3MBTL1 (0.40) L3MBTL1MCL1CTSSCTSLCTSB
SCHEMBL6181962 0.75 CTSS (0.50) L3MBTL1CTSSCTSLCTSBCTSK
SCHEMBL6565811 0.75 CTSS (0.40) CHRNB2CHRNB4CHRNA3CHRNA4MCL1
SCHEMBL6565044 0.73 CHRNB2 (0.41) CHRNB2CHRNB4CHRNA3CHRNA4L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed