SCHEMBL6563827

SCHEMBL6563827

CC(CCOC(=O)NCc1ccccc1)CC(=O)NCC#N

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 12/20 0.47
CTSL P07711 9/20 0.47
CTSB P07858 4/20 0.47
CTSK P43235 3/20 0.47
MCL1 Q07820 1/20 0.46
MEN1 O00255 1/20 0.43
HPGD P15428 1/20 0.43
KMT2A Q03164 1/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43
MAPT P10636 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PLA2G1B P04054 1/20 0.41
ATG4B Q9Y4P1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6567353 0.88 CHRNB2 (0.42) CTSSCTSLCTSBCTSKMCL1
SCHEMBL6565460 0.84 CHRNB2 (0.41) CTSSCTSLCTSBCTSKMCL1
SCHEMBL7456077 0.81 CTSS (0.57) CTSSCTSLCTSBCTSKL3MBTL1
SCHEMBL6181806 0.81 CTSS (0.57) CTSSCTSLCTSBCTSKL3MBTL1
SCHEMBL6565811 0.79 CTSS (0.40) CTSSCTSLCTSBCTSKMCL1
SCHEMBL6565044 0.78 CHRNB2 (0.41) CTSSCTSLCTSBCTSKHPGD
Hydrochloric Acid SCHEMBL28665674 0.75 CHRNB2 (0.50) MEN1KMT2ACHRNB2CHRNB4CHRNA3
SCHEMBL27558012 0.74 CHRNB2 (0.48) CHRNB2CHRNB4CHRNA3CHRNA4MAPT
SCHEMBL25990286 0.74 ALOX15 (0.55) MEN1KMT2ACHRNB2CHRNB4CHRNA3
SCHEMBL30805758 0.73 ALDH1A1 (0.58) MEN1HPGDKMT2AMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed