SCHEMBL6566818

SCHEMBL6566818

COc1ccc2c(c1)n(C(=O)O)c(=S)n2C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
ALDH1A1 P00352 2/20 0.45
HPGD P15428 2/20 0.45
HSD17B10 Q99714 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.42
AKR1C3 P42330 5/20 0.41
AKR1C2 P52895 5/20 0.41
PTGS2 P35354 3/20 0.41
TSHR P16473 3/20 0.41
PTGS1 P23219 2/20 0.41
CYP1A2 P05177 2/20 0.41
CDC42 P60953 1/20 0.41
RAC1 P63000 1/20 0.41
SLC22A6 Q4U2R8 1/20 0.41
GAA P10253 1/20 0.40
MAPT P10636 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
CA1 P00915 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6300235 0.80 NR1H2 (0.41) KDM4ESMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL7558266 0.71 GRM2 (0.44) KDM4ESMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL17422732 0.71 KDM4E (0.54) KDM4ESMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL8947431 0.70 HTR3A (0.56) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL7616142 0.70 HTR3A (0.45) KDM4ESMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL25184142 0.69 MTNR1A (0.49) KDM4ESMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL6740180 0.69 ALDH1A1 (0.45) KDM4ESMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL22261961 0.69 CCR9 (0.48) KDM4ESMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL25191837 0.68 MTNR1A (0.48) KDM4ESMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL20581381 0.67 MAOA (0.60) KDM4EAKR1C3AKR1C2PTGS2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268429-B1 VITRONECTIN RECEPTOR ANTAGONIST BICYCLIC COMPOUNDS, PREPARATION METHOD AND COMPOSITIONS CONTAINING SAME SERVIER LAB (FR) 2004-08-18 EP disclosed