SCHEMBL6567332

SCHEMBL6567332

CC(C)CCN(C#N)C(=O)C1(OC(=O)NCc2ccccc2)CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSB P07858 3/20 0.40
CTSS P25774 3/20 0.40
CTSL P07711 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
CTSK P43235 1/20 0.40
UTS2R Q9UKP6 2/20 0.38
MAPT P10636 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
ATM Q13315 1/20 0.35
GAA P10253 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
MCL1 Q07820 1/20 0.34
HPGD P15428 2/20 0.34
EPHX1 P07099 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRL1 P41146 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6567357 0.86 EPHX2 (0.40) CTSBCTSSCTSLKMT2AALDH1A1
SCHEMBL3898232 0.84 CTSB (0.43) CTSBCTSSCTSLCTSKATM
SCHEMBL3899355 0.78 HPGD (0.42) CTSBCTSSCTSLL3MBTL1MAPT
SCHEMBL3898239 0.76 CTSL (0.57) CTSBCTSSCTSLCTSKMCL1
SCHEMBL3892955 0.75 CTSL (0.42) CTSBCTSSCTSLL3MBTL1CTSK
SCHEMBL3908091 0.74 CTSS (0.41) CTSBCTSSCTSLCTSKHPGD
SCHEMBL7434373 0.74 CTSB (0.40) CTSBCTSSCTSLL3MBTL1CTSK
SCHEMBL6567349 0.73 CTSS (0.47) CTSBCTSSCTSLL3MBTL1CTSK
SCHEMBL3908088 0.73 CTSB (0.41) CTSBCTSSCTSLCTSKALDH1A1
SCHEMBL6565861 0.73 CTSB (0.36) CTSBCTSSCTSLL3MBTL1CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed