SCHEMBL6567357

SCHEMBL6567357

N#CN(CCCc1ccccc1)C(=O)C1(OC(=O)NCc2ccccc2)CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.40
CTSB P07858 2/20 0.38
CTSS P25774 2/20 0.38
CTSL P07711 1/20 0.37
EPHX1 P07099 3/20 0.36
BCHE P06276 1/20 0.36
MCL1 Q07820 1/20 0.36
HPGD P15428 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
ALDH1A1 P00352 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6567332 0.86 CTSB (0.40) CTSBCTSSCTSLEPHX1MCL1
SCHEMBL3898232 0.84 CTSB (0.43) CTSBCTSSCTSLEPHX1BCHE
SCHEMBL3899355 0.79 HPGD (0.42) CTSBCTSSCTSLEPHX1BCHE
SCHEMBL3898239 0.75 CTSL (0.57) CTSBCTSSCTSLEPHX1MCL1
SCHEMBL3908091 0.74 CTSS (0.41) CTSBCTSSCTSLHPGDOPRM1
SCHEMBL3902550 0.73 CTSC (0.45) CTSBCTSSCTSLALDH1A1
SCHEMBL7434373 0.73 CTSB (0.40) CTSBCTSSCTSLEPHX1MCL1
SCHEMBL3893533 0.73 CTSL (0.48) CTSBCTSSCTSLEPHX1MCL1
SCHEMBL6567042 0.73 CTSS (0.35) CTSBCTSSCTSLEPHX1BCHE
SCHEMBL3908088 0.73 CTSB (0.41) CTSBCTSSCTSLEPHX1MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed