SCHEMBL6568583

SCHEMBL6568583

O=C(Nc1ccc(OCc2ccccc2)cc1)Nc1cc(-c2nc3ccccc3s2)cc(Cl)c1O

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 11/20 0.58
EPHX2 P34913 11/20 0.58
MAPT P10636 7/20 0.50
TP53 P04637 3/20 0.50
ALOX5AP P20292 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
LMNA P02545 2/20 0.49
RXFP1 Q9HBX9 3/20 0.47
THRB P10828 1/20 0.47
MGLL Q99685 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6566878 0.87 MAPT (0.53) ALOX5EPHX2MAPTTP53SMN1; SMN2
SCHEMBL6524162 0.82 NAMPT (0.57) MAPTTP53SMN1; SMN2LMNAMGLL
SCHEMBL6519124 0.80 MAPT (0.47) MAPTTP53SMN1; SMN2LMNATHRB
SCHEMBL4350091 0.78 MAPT (0.53) MAPTTP53SMN1; SMN2LMNARXFP1
SCHEMBL13239642 0.77 ALOX5 (0.70) ALOX5EPHX2MAPTSMN1; SMN2LMNA
SCHEMBL4505884 0.77 TP53 (0.52) MAPTTP53SMN1; SMN2LMNATHRB
SCHEMBL6526530 0.76 MAPT (0.51) MAPTTP53SMN1; SMN2LMNATHRB
SCHEMBL6568636 0.75 KDM4E (0.49) MAPTTP53SMN1; SMN2LMNATHRB
SCHEMBL12470970 0.74 RAB9A (0.64) MAPTTP53SMN1; SMN2LMNA
SCHEMBL12846731 0.74 MAPT (0.50) MAPTTP53SMN1; SMN2LMNAMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed