SCHEMBL6568620

SCHEMBL6568620

Cc1c(Cl)cc(N(Cc2cc(Br)c(O)c(Br)c2)C(=O)NC(C)(C)C)c(O)c1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ANO1 Q5XXA6 3/20 0.33
POLB P06746 1/20 0.32
APEX1 P27695 1/20 0.32
CYP2C9 P11712 2/20 0.31
HSD17B10 Q99714 2/20 0.31
TSHR P16473 1/20 0.31
HIF1A Q16665 1/20 0.31
CYP2D6 P10635 1/20 0.31
KDM4E B2RXH2 3/20 0.31
MAPT P10636 2/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
TNF P01375 1/20 0.30
NOD2 Q9HC29 1/20 0.30
NOD1 Q9Y239 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6567254 0.89
SCHEMBL6568663 0.78 FAAH (0.39) POLBMAPTGAANPSR1TDP1
SCHEMBL6568607 0.68 POLB (0.35) CA1CA2POLBCYP2C9HSD17B10
SCHEMBL4357522 0.67 POLB (0.33) CA1CA2POLBCYP2C9HIF1A
SCHEMBL4344470 0.64 KMT2A (0.54) CA1CA2POLBAPEX1HSD17B10
SCHEMBL4345478 0.61 TSHR (0.47) APEX1HSD17B10TSHRMAPTGAA
SCHEMBL4353170 0.59 ALDH1A1 (0.36) POLBAPEX1MAPTGAANPSR1
SCHEMBL4350112 0.58 LMNA (0.33) POLBCYP2C9HSD17B10TSHRHIF1A
SCHEMBL4350106 0.58 POLB (0.52) POLBCYP2C9HIF1ACYP2D6KDM4E
SCHEMBL157575 0.58 CYP3A4 (0.44) CA1CA2CYP2C9HSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed