SCHEMBL6570778

SCHEMBL6570778

O=C(Cl)c1cc(Cl)c([N+](=O)[O-])cc1[N+](=O)[O-]

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 5/20 0.49
CYP3A4 P08684 2/20 0.49
ALDH1A1 P00352 1/20 0.49
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
GPR35 Q9HC97 2/20 0.44
SLC9A1 P19634 1/20 0.43
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
LMNA P02545 2/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
MMP8 P22894 1/20 0.40
MMP13 P45452 1/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8138894 0.90 VCAM1 (0.46) VCAM1CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL3328834 0.86 GPR35 (0.44) VCAM1CYP3A4ALDH1A1TSHRGPR35
SCHEMBL8575620 0.86 GPR35 (0.44) VCAM1CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL28515553 0.85 PPIA (0.42) VCAM1ALDH1A1TSHRMAPK1GPR35
SCHEMBL2977714 0.85 DTYMK (0.50) VCAM1CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL29596737 0.85 DTYMK (0.50) VCAM1CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL10562304 0.85 VCAM1 (0.49) VCAM1CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL3422244 0.83 CYP3A4 (0.57) VCAM1CYP3A4ALDH1A1TSHRMAPK1
SCHEMBL8142965 0.81 TSHR (0.43) CYP3A4ALDH1A1TSHRGPR35MAPT
SCHEMBL2924145 0.80 VCAM1 (0.45) VCAM1CYP3A4ALDH1A1TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0168733-A2 Process for the preparation of quinolinone and naphthyridoncarboxylic acids BAYER AG (DE) 1986-01-22 EP claimed
EP-1109550-B1 NOVEL NITROPHENYLAZIRIDINE COMPOUNDS AND THEIR USE AS PRODRUGS AUCKLAND UNISERVICES LTD (NZ) 2004-11-24 EP disclosed
US-6517836-B1 Aziridin-1-yl nitrobenzamides as prodrugs in conjunction with nitroreductase enzymes AUCKLAND UNISERVICES LIMITED (NZ) 2003-02-11 US disclosed
EP-1109550-A2 NOVEL NITROPHENYLAZIRIDINE COMPOUNDS AND THEIR USE AS PRODRUGS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2001-06-27 EP disclosed
WO-2000013683-A2 NOVEL NITROPHENYLAZIRIDINE COMPOUNDS AND THEIR USE AS PRODRUGS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-03-16 WO disclosed
EP-0689092-B1 Photographic elements containing development accelerators and release compounds that release development inhibitors EASTMAN KODAK CO (US) 1998-01-14 EP disclosed
EP-0684512-B1 Photographic elements containing release compounds EASTMAN KODAK CO (US) 1997-12-17 EP disclosed
EP-0684513-B1 Photographic elements containing development accelerators and release compounds that release development inhibitors EASTMAN KODAK CO (US) 1997-07-23 EP disclosed
US-5567577-A COMPRISING A BLOCKING GROUP FROM WHICH THE PHOTOGRAPHICALLY ACTIVE MOIETY IS RELEASED, A BALLASTING GROUP AND AN AQUEOUS SOLUBILIZING GROUP EASTMAN KODAK COMPANY (US) 1996-10-22 US disclosed
EP-0689092-A1 Photographic elements containing development accelerators and release compounds that release development inhibitors EASTMAN KODAK COMPANY (US) 1995-12-27 EP disclosed
US-5478711-A Photographic elements containing development accelerators and release compounds that release development inhibitors EASTMAN KODAK COMPANY (US) 1995-12-26 US disclosed
EP-0684513-A1 Photographic elements containing development accelerators and release compounds that release development inhibitors EASTMAN KODAK COMPANY (US) 1995-11-29 EP disclosed
EP-0684512-A1 Photographic elements containing release compounds EASTMAN KODAK COMPANY (US) 1995-11-29 EP disclosed
US-5460932-A Controlling color balance EASTMAN KODAK COMPANY (US) 1995-10-24 US disclosed
EP-0203488-A2 7-Azolyl-1-cyclopropyl-1,4-dihydro-4-oxo-3-quinoline carboxylic acids and 1,8-naphthyridine carboxylic acids, process for their preparation and bactericidal agents containing them BAYER AG (DE) 1986-12-03 EP disclosed
EP-0168733-A2 Process for the preparation of quinolinone and naphthyridoncarboxylic acids BAYER AG (DE) 1986-01-22 EP disclosed