SCHEMBL6570901

SCHEMBL6570901

[CH2]C(Cc1ccccc1)c1cccs1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
TSHR P16473 1/20 0.40
EPHX1 P07099 1/20 0.39
SLC5A2 P31639 1/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
KEAP1 Q14145 1/20 0.37
SLC6A2 P23975 3/20 0.36
TAAR1 Q96RJ0 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
MAOA P21397 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
CYP2A6 P11509 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6569435 0.80 TSHR (0.49) ALDH1A1TSHRNPC1RAB9AKMT2A
SCHEMBL3906596 0.78 SLC5A2 (0.52) ALDH1A1MAPTTSHREPHX1SLC5A2
SCHEMBL324034 0.78 CYP2C19 (0.48) ALDH1A1CES2CES1KEAP1SLC6A2
SCHEMBL30846613 0.77 EPHX1 (0.48) EPHX1SLC6A2TAAR1SLC6A4SLC6A3
SCHEMBL3289195 0.77 EPHX1 (0.48) EPHX1SLC6A2TAAR1SLC6A4SLC6A3
SCHEMBL30846601 0.77 EPHX1 (0.48) EPHX1SLC6A2TAAR1SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL9482622 0.76 EPHX1 (0.47) EPHX1SLC6A2TAAR1SLC6A4SLC6A3
SCHEMBL5647796 0.74 TRPA1 (0.43) ALDH1A1MAPTTSHREPHX1SLC5A2
SCHEMBL5651198 0.74 ANPEP (0.44) ALDH1A1MAPTTSHREPHX1SLC5A2
SCHEMBL5063737 0.74 CES2 (0.47) ALDH1A1MAPTTSHRCES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0328830-A1 4-Heteropentacyclic-4- N-(phenyl)amido piperidine compounds Ohmeda Pharmaceutical Products Division Inc. (US) 1989-08-23 EP claimed
CN-1178912-C Small molecule inhibitors of rotamase enzyme activity ������˹ҩƷ��˾ 2004-12-08 CN disclosed
CN-1542001-A Small molecule inhibitors of rotamase enzyme activity GPI����عɹ�˾ 2004-11-03 CN disclosed
EP-1404325-A2 METHOD FOR TREATING NERVE INJURY CAUSED BY SURGERY GUILFORD PHARMACEUTICALS INC. (US) 2004-04-07 EP disclosed
WO-2002096420-A2 METHOD FOR TREATING NERVE INJURY CAUSED BY SURGERY GUILFORD PHARMACEUTICALS INC. (US) 2002-12-05 WO disclosed
CN-1336930-A Bridged heterocyclic derivatives GPINIL HOLDING CORP (US) 2002-02-20 CN disclosed
EP-1127049-A1 BRIDGED HETEROCYCLIC DERIVATIVES GPI NIL Holdings, Inc. (US) 2001-08-29 EP disclosed
EP-1011650-A1 METHOD FOR PREVENTING AND TREATING HEARING LOSS USING SENSORINEUROTROPHIC COMPOUNDS Amgen Inc., (US) 2000-06-28 EP disclosed
WO-2000016603-A2 BRIDGED HETEROCYCLIC DERIVATIVES GPI NIL HOLDINGS, INC. (US) 2000-03-30 WO disclosed
WO-1999014998-A2 METHOD FOR PREVENTING AND TREATING HEARING LOSS USING SENSORINEUROTROPHIC COMPOUNDS AMGEN INC. (US) 1999-04-01 WO disclosed
CN-1187188-A Small molecule inhibitors of rotamase enzyme activity GUILFORD PHARM INC (US) 1998-07-08 CN disclosed