SCHEMBL6570967

SCHEMBL6570967

COc1ccc(-c2cc(N(CCO)CCO)ccc2N)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RELA Q04206 2/20 0.38
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
USP8 P40818 1/20 0.37
ABL1 P00519 1/20 0.37
ABCB1 P08183 1/20 0.37
BCR P11274 1/20 0.37
MAPT P10636 3/20 0.37
BACE1 P56817 2/20 0.37
PRUNE1 Q86TP1 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
IKBKB O14920 1/20 0.37
ADORA3 P0DMS8 1/20 0.36
RPS6KA3 P51812 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ADK P55263 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6572323 0.87 ALOX15 (0.40) RELAABL1ABCB1BCRMAPT
SCHEMBL6574721 0.87 TDO2 (0.42) ABL1MAPTRPS6KA3ALDH1A1HSD17B10
SCHEMBL6572855 0.84 ALDH1A1 (0.42) RELAMAPTMEN1KMT2ACYP3A4
SCHEMBL6572316 0.84 S100B (0.40) USP8MAPTBACE1SMN1; SMN2RPS6KA3
SCHEMBL6572518 0.84 MAPT (0.38) MAPTSMN1; SMN2IKBKBADKMEN1
SCHEMBL6571892 0.83 MAPT (0.37) USP8MAPTSMN1; SMN2KDM4EMEN1
SCHEMBL6572200 0.82 USP7 (0.40) USP8ABL1ABCB1BCRMAPT
SCHEMBL6574636 0.82 KMT2A (0.42) RELAMAPTSMN1; SMN2IKBKBCYP1A2
SCHEMBL6571136 0.82 DYRK1A (0.41) RELAMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL6571049 0.81 KMT2A (0.35) USP8MAPTSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed