SCHEMBL6572844

SCHEMBL6572844

CNc1ccc(N)c(-c2cccc(OC)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.48
ALDH1A1 P00352 4/20 0.45
HSD17B10 Q99714 4/20 0.45
LMNA P02545 3/20 0.45
MAPT P10636 1/20 0.45
ADORA2A P29274 2/20 0.44
ADORA1 P30542 1/20 0.44
CYP3A4 P08684 5/20 0.43
HDAC2 Q92769 1/20 0.43
TGFBR2 P37173 1/20 0.42
KDM4E B2RXH2 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP1A2 P05177 4/20 0.41
CYP2D6 P10635 4/20 0.41
CYP2C19 P33261 4/20 0.41
CLK4 Q9HAZ1 3/20 0.41
MAPK1 P28482 2/20 0.41
CYP2C9 P11712 2/20 0.41
ALOX15 P16050 1/20 0.41
CYP1A1 P04798 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28255761 0.84 TDO2 (0.55) TDO2ALDH1A1HSD17B10LMNAMAPT
SCHEMBL6572471 0.83 NR4A1 (0.44) ALDH1A1HSD17B10MAPTCYP3A4HDAC2
SCHEMBL6570805 0.81 CYP1A2 (0.46) TDO2ALDH1A1HSD17B10LMNAMAPT
SCHEMBL6573720 0.81 MEN1 (0.46) TDO2ALDH1A1HSD17B10LMNAMAPT
SCHEMBL3789189 0.81 MAP4K4 (0.46) MAPTCYP3A4KITCNR1MAOB
SCHEMBL6571024 0.81 CYP3A4 (0.58) TDO2ALDH1A1HSD17B10LMNAMAPT
Hydrochloric Acid SCHEMBL6570983 0.80 ALDH1A1 (0.56) TDO2ALDH1A1HSD17B10LMNAMAPT
SCHEMBL3788714 0.79 ALDH1A1 (0.48) TDO2ALDH1A1HSD17B10HDAC2KMT2A
SCHEMBL6572598 0.78 ALDH1A1 (0.59) TDO2ALDH1A1HSD17B10LMNAMAPT
SCHEMBL6572177 0.78 HSD17B1 (0.41) ALDH1A1ADORA2AADORA1CYP3A4CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed