SCHEMBL6572471

SCHEMBL6572471

CNc1ccc(N)c(-c2ccc(OC)cc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A1 P22736 1/20 0.44
MAPT P10636 5/20 0.42
GAA P10253 4/20 0.42
TDP1 Q9NUW8 4/20 0.42
KDM4E B2RXH2 3/20 0.42
RAB9A P51151 3/20 0.42
THRB P10828 2/20 0.42
RECQL P46063 2/20 0.42
MAPK1 P28482 2/20 0.42
NPC1 O15118 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
APP P05067 2/20 0.42
ABL1 P00519 1/20 0.42
ABCB1 P08183 1/20 0.42
BCR P11274 1/20 0.42
ALDH1A1 P00352 4/20 0.41
HTT P42858 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6572844 0.83 TDO2 (0.48) MAPTKDM4EMAPK1ALDH1A1KMT2A
SCHEMBL3790061 0.82 HTR6 (0.39) NR4A1MAPTTDP1KDM4ERAB9A
SCHEMBL6570748 0.81 TDP1 (0.39) MAPTGAATDP1KDM4ERAB9A
SCHEMBL6572389 0.80 GAA (0.49) NR4A1MAPTGAAKDM4ERAB9A
SCHEMBL6571911 0.80 ALDH1A1 (0.49) NR4A1MAPTGAAKDM4ETHRB
SCHEMBL6573189 0.79 CYP3A4 (0.38) TDP1KDM4ERAB9AMAPK1NPC1
SCHEMBL6571412 0.79 APP (0.47) MAPTGAATDP1KDM4ETHRB
SCHEMBL7690453 0.79 CA1 (0.49) MAPTABL1ABCB1BCRALDH1A1
SCHEMBL6572041 0.79 GAA (0.47) NR4A1MAPTGAATDP1KDM4E
SCHEMBL453782 0.79 TDP1 (0.56) NR4A1MAPTTDP1KDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed