SCHEMBL6573189

SCHEMBL6573189

CNc1ccc(N)c(-c2ccc(Cl)cc2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.38
ALDH1A1 P00352 4/20 0.38
TSHR P16473 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
ALOX15 P16050 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
IKBKB O14920 1/20 0.37
CHUK O15111 1/20 0.37
KIF11 P52732 1/20 0.37
APP P05067 1/20 0.36
AHR P35869 1/20 0.36
TDO2 P48775 1/20 0.36
IDO1 P14902 4/20 0.36
MAP4K4 O95819 3/20 0.36
KDM4E B2RXH2 2/20 0.36
HPGD P15428 1/20 0.36
PPARG P37231 1/20 0.36
STAT3 P40763 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3790061 0.85 HTR6 (0.39) CYP3A4ALDH1A1TSHRTDP1ALOX15
SCHEMBL6570748 0.84 TDP1 (0.39) CYP3A4ALDH1A1TSHRTDP1ALOX15
SCHEMBL1577931 0.82 TSHR (0.54) CYP3A4ALDH1A1TSHRTDP1ALOX15
SCHEMBL6571412 0.82 APP (0.47) CYP3A4ALDH1A1TDP1ALOX15APP
SCHEMBL3788714 0.81 ALDH1A1 (0.48) ALDH1A1TSHRTDP1IKBKBCHUK
SCHEMBL14907071 0.80 TSHR (0.56) CYP3A4ALDH1A1TSHRTDP1ALOX15
SCHEMBL6574394 0.79 MAPT (0.40) CYP3A4ALDH1A1TSHRTDP1ALOX15
SCHEMBL6572471 0.79 NR4A1 (0.44) CYP3A4ALDH1A1TSHRTDP1APP
SCHEMBL1578529 0.79 HDAC1 (0.50) ALDH1A1TDP1SMN1; SMN2KDM4EHPGD
SCHEMBL6570788 0.78 KIF11 (0.61) ALDH1A1KIF11APPKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed