SCHEMBL6573199

SCHEMBL6573199

Cc1cc(C)c(N)c(-c2cc(N)ccc2N)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 3/20 0.43
PDE10A Q9Y233 1/20 0.41
ALDH1A1 P00352 9/20 0.40
PLA2G7 Q13093 1/20 0.37
TSHR P16473 4/20 0.36
KDM4E B2RXH2 4/20 0.36
CYP3A4 P08684 3/20 0.36
GAA P10253 3/20 0.36
MAPT P10636 3/20 0.36
LMNA P02545 1/20 0.36
RAPGEF4 Q8WZA2 1/20 0.36
TDP1 Q9NUW8 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
TP53 P04637 1/20 0.35
THRB P10828 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 3/20 0.35
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
CASP7 P55210 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23932622 0.81 KDM4E (0.48) ALDH1A1TSHRKDM4ECYP3A4GAA
SCHEMBL6711282 0.80 CASP1 (0.46) CASP1PDE10AALDH1A1PLA2G7TSHR
SCHEMBL6572820 0.78 CYP3A4 (0.41) CASP1PDE10AALDH1A1PLA2G7TSHR
SCHEMBL7684845 0.78 ALDH1A1 (0.50) CASP1PDE10AALDH1A1PLA2G7TSHR
SCHEMBL3789931 0.78 ALDH1A1 (0.52) ALDH1A1KDM4ECYP3A4GAAMAPT
Hydrochloric Acid SCHEMBL6572317 0.77 PLA2G7 (0.49) CASP1PDE10AALDH1A1PLA2G7TSHR
Hydrochloric Acid SCHEMBL6574671 0.77 ALDH1A1 (0.46) CASP1PDE10AALDH1A1PLA2G7TSHR
SCHEMBL3791658 0.76 ACHE (0.42) CASP1PDE10AALDH1A1TSHRKDM4E
SCHEMBL3338155 0.76 CASP1 (0.46) CASP1PDE10AALDH1A1TSHRCYP3A4
SCHEMBL28543486 0.75 CASP1 (0.44) CASP1PDE10AALDH1A1PLA2G7TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed