SCHEMBL6574728

SCHEMBL6574728

COCCN(CCOC)c1ccc(N)c(-c2ccc(Cl)cc2)c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
CRHR1 P34998 7/20 0.37
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
ATM Q13315 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CYP3A4 P08684 1/20 0.34
DPP4 P27487 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ADK P55263 1/20 0.34
LIMK1 P53667 1/20 0.34
S100B P04271 1/20 0.33
F2 P00734 1/20 0.32
PRSS1 P07477 1/20 0.32
PRSS2 P07478 1/20 0.32
PRSS3 P35030 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6572811 0.89 CRHR1 (0.37) KMT2AMEN1CRHR1CYP3A4DPP4
SCHEMBL6571429 0.89 ALDH1A1 (0.36) KMT2AMEN1SMN1; SMN2TP53CYP3A4
SCHEMBL6570799 0.87 GRM2 (0.38) SMN1; SMN2RAB9AS100BF2PRSS1
SCHEMBL6570859 0.87 S100B (0.37) KMT2AMEN1CRHR1SMN1; SMN2LMNA
SCHEMBL6572008 0.87 MAPT (0.35) CRHR1LMNATP53CYP3A4RAB9A
SCHEMBL6571313 0.87 FYN (0.38) KMT2AMEN1CRHR1CYP3A4
SCHEMBL6571876 0.86 CYP3A4 (0.40) KMT2AMEN1CRHR1LMNACYP3A4
SCHEMBL6571984 0.86 S100B (0.36) KMT2AMEN1CRHR1SMN1; SMN2ATM
SCHEMBL6572323 0.86 ALOX15 (0.40) KMT2ACRHR1CYP3A4ADK
SCHEMBL6571056 0.86 MGAM (0.36) KMT2AMEN1S100BF2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed