SCHEMBL6574930

SCHEMBL6574930

NC(N)(N)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
CA1 P00915 4/20 0.55
CA2 P00918 4/20 0.55
CA9 Q16790 3/20 0.55
CA5A P35218 2/20 0.55
CA12 O43570 2/20 0.50
CA14 Q9ULX7 2/20 0.50
HSD17B10 Q99714 2/20 0.50
LOXL2 Q9Y4K0 1/20 0.50
ACHE P22303 1/20 0.50
CA3 P07451 1/20 0.50
CA4 P22748 1/20 0.50
CA6 P23280 1/20 0.50
CA7 P43166 1/20 0.50
CA13 Q8N1Q1 1/20 0.50
CA5B Q9Y2D0 1/20 0.50
TSHR P16473 1/20 0.48
APP P05067 1/20 0.48
LMNA P02545 1/20 0.48
CES1 P23141 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3154297 0.82 ALDH1A1 (0.52) ALDH1A1CA1CA2CA9CA5A
Hydrochloric Acid SCHEMBL3928206 0.80 ALDH1A1 (0.50) ALDH1A1CA1CA2CA9CA5A
SCHEMBL9003264 0.80 LOXL2 (0.55) ALDH1A1CA1CA2CA9CA5A
SCHEMBL1682720 0.80 ALDH1A1 (0.54) ALDH1A1CA1CA2CA9CA5A
Hydrazine SCHEMBL27401571 0.79 ALDH1A1 (0.74) ALDH1A1CA1CA2CA9CA5A
SCHEMBL27909482 0.79 ALDH1A1 (0.72) ALDH1A1CA1CA2CA9CA5A
SCHEMBL22567 0.79 ALDH1A1 (0.72) ALDH1A1CA1CA2CA9CA5A
SCHEMBL5684191 0.79 HSD11B1 (0.53) ALDH1A1CA1CA2CA9CA5A
SCHEMBL5180046 0.78 ALDH1A1 (0.52) ALDH1A1CA1CA2CA9CA5A
SCHEMBL445417 0.77 CA1 (0.56) ALDH1A1CA1CA2CA9CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785928-B1 NOVEL N3 S2 CHELATING LIGANDS OPTIONALLY RADIOLABELLED WITH Tc OR Re, USEFUL FOR DIAGNOSTIC OR THERAPEUTIC APPLICATIONS MERCK FROSST CANADA INC (CA) 2004-04-28 EP disclosed
EP-0785951-B1 TC OR RE RADIOLABELLED SOMATOSTATIN ANALOGS MERCK FROSST CANADA INC (CA) 2002-04-24 EP disclosed
EP-0785928-A1 NOVEL N3 S2 CHELATING LIGANDS OPTIONALLY RADIOLABELLED WITH Tc OR Re, USEFUL FOR DIAGNOSTIC OR THERAPEUTIC APPLICATIONS MERCK FROSST CANADA INC. (CA) 1997-07-30 EP disclosed
US-5632969-A N3 S2 chelating ligands optionally radiolabelled with Tc or Re, useful for diagnostic or therapeutic applications MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5556939-A TC or RE radionuclide labelled chelate, hexapeptide complexes useful for diagnostic or therapeutic applications MERCK FROSST CANADA, INC. (CA) 1996-09-17 US disclosed
US-5539138-A High affinity chelates containing isothiocyanate groups, useful for coupling with peptides and proteins MERCK FROSST CANADA, INC. (CA) 1996-07-23 US disclosed
WO-1996011918-A1 NOVEL N3S2 CHELATING LIGANDS OPTIONALLY RADIOLABELLED WITH Tc OR Re, USEFUL FOR DIAGNOSTIC OR THERAPEUTIC APPLICATIONS MERCK FROSST CANADA INC. (CA) 1996-04-25 WO disclosed