SCHEMBL6575713

SCHEMBL6575713

Cc1ccc(N2C(=O)CCc3ccc(O)cc32)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.46
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 2/20 0.41
F2 P00734 1/20 0.41
ELANE P08246 1/20 0.41
CTSG P08311 1/20 0.41
CMA1 P23946 1/20 0.41
CTRC Q99895 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
MIF P14174 1/20 0.40
GAA P10253 3/20 0.39
MEN1 O00255 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PBRM1 Q86U86 1/20 0.39
MAPT P10636 1/20 0.39
MGLL Q99685 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12559590 0.79 L3MBTL1 (0.54) KMT2ANPC1RAB9AALDH1A1LMNA
SCHEMBL5215688 0.78 HPGD (0.53) KMT2ANPC1RAB9AALDH1A1LMNA
SCHEMBL5817493 0.78 MGLL (0.43) KMT2ANPC1RAB9AALDH1A1LMNA
SCHEMBL8613287 0.76 MAPT (0.39) KMT2AALDH1A1LMNAF2ELANE
SCHEMBL11692973 0.75 KMT2A (0.56) KMT2AESR1GAAMEN1SMN1; SMN2
SCHEMBL1949985 0.75 LMNA (0.64) KMT2AALDH1A1LMNAF2ELANE
SCHEMBL29846831 0.74 PBRM1 (0.46) ESR1ESR2PBRM1
SCHEMBL6073803 0.74 PBRM1 (0.46) ESR1ESR2PBRM1
SCHEMBL3431666 0.74 DRD2 (0.44) KMT2ANPC1RAB9AALDH1A1L3MBTL1
SCHEMBL5218324 0.73 SLC6A2 (0.50) KMT2AALDH1A1LMNAF2ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0937045-B1 N-ARYL SUBSTITUTED TETRAHYDROQUINOLINES LIGANDS FOR RETINOID RECEPTORS HAVING AGONIST, ANTAGONIST OR INVERSE AGONIST TYPE ACTIVITY ALLERGAN INC (US) 2004-04-28 EP disclosed