SCHEMBL6578008

SCHEMBL6578008

CC1(C)CCN(c2ccccc2)c2cc(C#Cc3ccccc3)ccc21

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RARB P10826 7/20 0.51
RARG P13631 7/20 0.51
RARA P10276 5/20 0.51
CYP26A1 O43174 1/20 0.43
CYP3A4 P08684 1/20 0.43
CRABP2 P29373 1/20 0.43
GRM5 P41594 10/20 0.42
SRD5A1 P18405 2/20 0.39
SRD5A2 P31213 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6574370 0.89 RARB (0.67) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8616759 0.87 RARB (0.42) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6578033 0.86 RARA (0.40) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8614817 0.83 RARB (0.52) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6578025 0.80 RARB (0.65) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6574407 0.79 HSD11B1 (0.42) RARBRARGRARACYP3A4
SCHEMBL6575676 0.76 RARB (0.39) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6574397 0.75 RARA (0.37) RARBRARGRARA
SCHEMBL20061936 0.74 HSD11B1 (0.38) RARBRARGCYP3A4
SCHEMBL6576434 0.74 RARB (0.48) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0937045-B1 N-ARYL SUBSTITUTED TETRAHYDROQUINOLINES LIGANDS FOR RETINOID RECEPTORS HAVING AGONIST, ANTAGONIST OR INVERSE AGONIST TYPE ACTIVITY ALLERGAN INC (US) 2004-04-28 EP disclosed