SCHEMBL6578586

SCHEMBL6578586

[CH2]c1cccc(-c2n[nH]c(-c3ccc(OCF)c(F)c3)n2)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.44
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
NR1H2 P55055 3/20 0.40
NR1H3 Q13133 3/20 0.40
ATAD2 Q6PL18 1/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
DGAT1 O75907 1/20 0.39
LCK P06239 1/20 0.37
BTK Q06187 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581499 0.86 NR1H2 (0.50) S1PR1ADORA2AADORA1NR1H2NR1H3
SCHEMBL6582892 0.84 ADORA2A (0.41) S1PR1ADORA2AADORA1NR1H2NR1H3
SCHEMBL6579126 0.83 NR1H2 (0.49) S1PR1ADORA2AADORA1NR1H2NR1H3
SCHEMBL6578288 0.82 S1PR1 (0.47) S1PR1ADORA2AADORA1NR1H2NR1H3
Hydrochloric Acid SCHEMBL6578720 0.81 S1PR1 (0.46) S1PR1ADORA2AADORA1NR1H2NR1H3
SCHEMBL6581439 0.76 NR1H2 (0.52) ADORA2AADORA1NR1H2NR1H3ATAD2
Hydrochloric Acid SCHEMBL6581197 0.72 S1PR1 (0.53) S1PR1ADORA2AADORA1NR1H2NR1H3
SCHEMBL6578742 0.72 NR1H2 (0.67) S1PR1ADORA2AADORA1NR1H2NR1H3
SCHEMBL6580942 0.70 HTR7 (0.46) S1PR1ADORA2AADORA1NR1H2NR1H3
Hydrochloric Acid SCHEMBL6581027 0.70 HTR7 (0.46) S1PR1ADORA2AADORA1NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP claimed