SCHEMBL6578631

SCHEMBL6578631

CCCCCN1CCCC2CC=CC=C21

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 7/20 0.33
DRD4 P21917 7/20 0.33
DRD5 P21918 7/20 0.33
DRD3 P35462 7/20 0.33
HTR1A P08908 6/20 0.33
KCNH2 Q12809 1/20 0.33
BCHE P06276 1/20 0.33
GNAI3 P08754 1/20 0.33
GNAO1 P09471 1/20 0.33
GNAI1 P63096 1/20 0.33
DRD2 P14416 6/20 0.33
LTA4H P09960 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11660093 0.96 DRD2 (0.33) DRD1DRD4DRD5DRD3HTR1A
SCHEMBL11390969 0.91 HTR1A (0.37) DRD1DRD4DRD5DRD3HTR1A
SCHEMBL11440182 0.90 DRD2 (0.38) DRD1DRD4DRD5DRD3DRD2
SCHEMBL11789421 0.83 DRD2 (0.30) DRD1DRD4DRD5DRD3DRD2
SCHEMBL9355576 0.81 SLC18A3 (0.31)
SCHEMBL23047083 0.75
SCHEMBL4674255 0.75
SCHEMBL9664096 0.74
SCHEMBL9637964 0.72 HTR1A (0.34) DRD1DRD4DRD5DRD3HTR1A
SCHEMBL8564164 0.72 MGLL (0.43) DRD4DRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0937045-B1 N-ARYL SUBSTITUTED TETRAHYDROQUINOLINES LIGANDS FOR RETINOID RECEPTORS HAVING AGONIST, ANTAGONIST OR INVERSE AGONIST TYPE ACTIVITY ALLERGAN INC (US) 2004-04-28 EP disclosed
US-5739338-A SKIN DISORDERS, ANTIINFLAMMATORY AGENTS, ANTITUMOR AGENTS, VISION DEFECTS, VIRICIDES, IMMUNOSUPPRESSANTS ALLERGAN (US) 1998-04-14 US disclosed
US-4111929-A POLYACRYLONITRILE IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1978-09-05 US disclosed