SCHEMBL6579923

SCHEMBL6579923

COc1cccc(-c2nc(OCCCCl)ns2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.51
MAPT P10636 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
KDM4E B2RXH2 1/20 0.50
LMNA P02545 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.44
NFKB1 P19838 1/20 0.44
RAB9A P51151 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
ALDH1A1 P00352 1/20 0.42
DYRK1A Q13627 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
DCTPP1 Q9H773 2/20 0.41
PTPN1 P18031 1/20 0.41
SREBF2 Q12772 1/20 0.41
TLR7 Q9NYK1 1/20 0.39
USP2 O75604 1/20 0.39
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581805 0.82 HSD17B1 (0.55) CYP19A1LMNASMN1; SMN2NFKB1RAB9A
SCHEMBL6581716 0.81 ADORA3 (0.46) MAPTKDM4ESMN1; SMN2RAB9AALDH1A1
SCHEMBL8838312 0.78 CYP19A1 (0.49) CYP19A1MAPTTDP1KDM4ELMNA
SCHEMBL8715461 0.76 CYP19A1 (0.59) CYP19A1MAPTTDP1KDM4ELMNA
SCHEMBL6581800 0.76 CYP3A4 (0.48) CYP19A1MAPTTDP1KDM4ELMNA
Hydrochloric Acid SCHEMBL6581834 0.76 BLM (0.49) MAPTTDP1KDM4ELMNASMN1; SMN2
SCHEMBL8838311 0.74 CYP19A1 (0.48) CYP19A1MAPTTDP1KDM4ELMNA
SCHEMBL29673242 0.74 CYP19A1 (0.59) CYP19A1MAPTTDP1KDM4ELMNA
SCHEMBL20588052 0.74 CYP19A1 (0.59) CYP19A1MAPTTDP1KDM4ELMNA
SCHEMBL6581534 0.74 CYP19A1 (0.59) CYP19A1MAPTTDP1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737680-B1 (Phenylalkylaminoalkyloxyl)-hetero-aryl compounds, processes and intermediates for their preparation and medicaments containing these compounds SOLVAY PHARM GMBH (DE) 2004-03-03 EP disclosed
US-5679699-A ANTIISCHEMIC AGENTS, HEART RATE LOWERING AGENTS KALI-CHEMIE PHARMA GMBH (DE) 1997-10-21 US disclosed
EP-0737680-A1 (Phenylalkylaminoalkyloxyl)-hetero-aryl compounds, processes and intermediates for their preparation and medicaments containing these compounds Kali-Chemie Pharma GmbH (DE) 1996-10-16 EP disclosed
US-5547967-A HYPOTENSIVE AGENT, ANTIISCHEMIC AGENT KALI-CHEMIE PHARMA GMBH (DE) 1996-08-20 US disclosed