SCHEMBL6581534

SCHEMBL6581534

COc1cccc(-c2nc(O)ns2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.59
MAPT P10636 2/20 0.51
TDP1 Q9NUW8 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
NFKB1 P19838 1/20 0.51
RAB9A P51151 1/20 0.51
NFKB2 Q00653 1/20 0.51
RELA Q04206 1/20 0.51
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 2/20 0.48
LMNA P02545 1/20 0.48
HSD17B1 P14061 2/20 0.46
HSD17B2 P37059 2/20 0.46
HDAC4 P56524 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
DYRK1A Q13627 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
TRPM8 Q7Z2W7 1/20 0.44
USP2 O75604 2/20 0.44
HSD17B10 Q99714 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20588052 0.81 CYP19A1 (0.59) CYP19A1MAPTTDP1SMN1; SMN2NFKB1
SCHEMBL8715461 0.81 CYP19A1 (0.59) CYP19A1MAPTTDP1SMN1; SMN2NFKB1
SCHEMBL29673242 0.81 CYP19A1 (0.59) CYP19A1MAPTTDP1SMN1; SMN2NFKB1
SCHEMBL28406603 0.80 CYP19A1 (0.73) CYP19A1MAPTTDP1SMN1; SMN2NFKB1
SCHEMBL30287350 0.80 CYP19A1 (0.73) CYP19A1MAPTTDP1SMN1; SMN2NFKB1
SCHEMBL6581811 0.74 ADORA3 (0.59) MAPTSMN1; SMN2RAB9AALDH1A1KDM4E
SCHEMBL8838311 0.74 CYP19A1 (0.48) CYP19A1MAPTTDP1SMN1; SMN2NFKB1
SCHEMBL6579923 0.74 CYP19A1 (0.51) CYP19A1MAPTTDP1SMN1; SMN2NFKB1
SCHEMBL1180747 0.73 RAB9A (0.59) MAPTTDP1SMN1; SMN2NFKB1RAB9A
SCHEMBL1180755 0.73 HSD17B1 (0.74) CYP19A1MAPTSMN1; SMN2RAB9AHSD17B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737680-B1 (Phenylalkylaminoalkyloxyl)-hetero-aryl compounds, processes and intermediates for their preparation and medicaments containing these compounds SOLVAY PHARM GMBH (DE) 2004-03-03 EP disclosed
EP-0737680-A1 (Phenylalkylaminoalkyloxyl)-hetero-aryl compounds, processes and intermediates for their preparation and medicaments containing these compounds Kali-Chemie Pharma GmbH (DE) 1996-10-16 EP disclosed