SCHEMBL6580736

SCHEMBL6580736

Fc1ccc(-n2cc(C3=CCNCC3)c3cc(Cl)ccc32)cc1

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 12/20 0.61
KCNH2 Q12809 5/20 0.57
HTR1A P08908 1/20 0.48
DRD2 P14416 1/20 0.48
HTR2A P28223 1/20 0.48
HTR7 P34969 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27751697 1.00 HTR6 (0.61) HTR6KCNH2HTR1ADRD2HTR2A
SCHEMBL9147029 0.91 HTR6 (0.56) HTR6KCNH2
SCHEMBL9462735 0.91 HTR6 (0.68) HTR6KCNH2HTR1AHTR2AHTR7
SCHEMBL9150425 0.87 HTR6 (0.55) HTR6KCNH2HTR1AHTR2A
SCHEMBL9462566 0.85 HTR6 (0.56) HTR6KCNH2HTR1A
SCHEMBL10874677 0.83 HTR6 (0.57) HTR6HTR1AHTR2AHTR7
SCHEMBL7685212 0.82 HTR6 (0.52) HTR6HTR1ADRD2HTR2AHTR7
SCHEMBL9463173 0.82 HTR6 (0.61) HTR6KCNH2HTR1AHTR2A
SCHEMBL6583508 0.81 HTR6 (0.54) HTR6KCNH2HTR1A
SCHEMBL9149499 0.80 HTR6 (0.52) HTR6HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1243001-C Process for the manufacture of sertindole LUNDBECK & CO AS H (DK) 2006-02-22 CN claimed
EP-1260511-B1 Process for the preparation of 5-chloro-1-(4-fluorophenyl)-3-(1,2,3,6-tetrahydropyridin-4-yl)indole and method of manufacturing sertindole LUNDBECK & CO AS H (DK) 2004-12-29 EP claimed
EP-0983264-B1 METHOD OF MANUFACTURING SERTINDOLE LUNDBECK & CO AS H (DK) 2004-02-04 EP claimed
EP-1260511-A1 Process for the preparation of 5-chloro-1-(4-fluorophenyl)-3-(1,2,3,6-tetrahydropyridin-4-yl)indole and method of manufacturing sertindole H. Lundbeck A/S (DK) 2002-11-27 EP claimed
US-6335463-B1 Method of manufacturing sertindole H. LUNDBECK A/S (DK) 2002-01-01 US claimed
CN-1261363-A Process for the manufacture of sertindole LUNDBECK & CO AS H (DK) 2000-07-26 CN claimed
EP-0983264-A1 METHOD OF MANUFACTURING SERTINDOLE H. LUNDBECK A/S (DK) 2000-03-08 EP claimed
WO-1998051685-A1 METHOD OF MANUFACTURING SERTINDOLE H. LUNDBECK A/S (DK) 1998-11-19 WO claimed
CN-101899036-B Method for preparing sertindole by using alkyl imidazole type ionic liquid as solvent UNIV ZHENGZHOU 2012-12-19 CN disclosed
CN-101899036-A Method for preparing sertindole by using alkyl imidazole type ionic liquid as solvent UNIV ZHENGZHOU 2010-12-01 CN disclosed
CN-101362749-A Sertindole synthesis method SHANGHAI INST PHARM INDUSTRY (CN) 2009-02-11 CN disclosed
CN-1301963-C Process for producing N-(4-fluobenzene radical)-N-(2-hydroxy-4-chlorobenzene group) glycocoll LUNDBECK & CO AS H (DK) 2007-02-28 CN disclosed
CN-1243001-C Process for the manufacture of sertindole LUNDBECK & CO AS H (DK) 2006-02-22 CN disclosed
CN-1243001-C Process for the manufacture of sertindole LUNDBECK & CO AS H (DK) 2006-02-22 CN disclosed
WO-1998051685-A1 METHOD OF MANUFACTURING SERTINDOLE H. LUNDBECK A/S (DK) 1998-11-19 WO disclosed
WO-1998051685-A1 METHOD OF MANUFACTURING SERTINDOLE H. LUNDBECK A/S (DK) 1998-11-19 WO disclosed
US-RE34299-E Psychological disorders, neuroleptic agents, analgesics H. LUNDBECK A/S (DK) 1993-06-29 US disclosed
EP-0200322-B1 HETEROCYCLIC COMPOUNDS H. LUNDBECK A/S (DK) 1990-02-28 EP disclosed
US-4710500-A 1-(4'-fluorophenyl)-3,5-substituted indoles useful in the treatment of psychic disorders and pharmaceutical compositions thereof H. LUNDBECK A/S (DK) 1987-12-01 US disclosed
EP-0200322-A1 Heterocyclic compounds H. LUNDBECK A/S (DK) 1986-11-05 EP disclosed