SCHEMBL6581464

SCHEMBL6581464

Cc1ccc2cc(OCc3c(C)ccc(N)c3C)ccc2n1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
CASP6 P55212 1/20 0.44
ALDH1A1 P00352 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NCF1 P14598 10/20 0.41
CYP1A2 P05177 1/20 0.40
RAB9A P51151 2/20 0.39
MAPT P10636 2/20 0.39
NPC1 O15118 1/20 0.39
HTT P42858 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TEC P42680 1/20 0.37
MAOB P27338 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6936592 0.80 KDM4E (0.42) KDM4ELMNAPOLBCASP6ALDH1A1
SCHEMBL6581453 0.80 ALDH1A1 (0.40) LMNAALDH1A1CYP1A2RAB9AMAPT
SCHEMBL6580627 0.78 NCF1 (0.41) KDM4ELMNAPOLBCASP6ALDH1A1
SCHEMBL6578833 0.77 NCF1 (0.40) KDM4ELMNAPOLBCASP6ALDH1A1
SCHEMBL6580770 0.77 NCF1 (0.40) KDM4ELMNAPOLBCASP6ALDH1A1
SCHEMBL6578780 0.77 NCF1 (0.40) KDM4ELMNAPOLBCASP6ALDH1A1
SCHEMBL6578484 0.76 NCF1 (0.39) KDM4ELMNAPOLBCASP6ALDH1A1
SCHEMBL6576073 0.76 KDM4E (0.38) KDM4ELMNAPOLBCASP6ALDH1A1
SCHEMBL6578390 0.75 NQO1 (0.41) KDM4ELMNAPOLBCASP6ALDH1A1
SCHEMBL6581525 0.74 NCF1 (0.39) KDM4ELMNAPOLBCASP6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0867432-B1 Fused N-heterocyclic compounds substituted with benzyloxy, process for their preparation and their use as bradykinin receptor antagonists AVENTIS PHARMA GMBH (DE) 2004-06-09 EP disclosed
EP-0867432-A2 Fused N-heterocyclic compounds substituted with benzyloxy, process for their preparation and their use as bradykinin receptor antagonists HOECHST AKTIENGESELLSCHAFT (DE) 1998-09-30 EP disclosed