SCHEMBL6582224

SCHEMBL6582224

CC(C)C=CN1CCOCC1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.39
ALDH1A1 P00352 5/20 0.37
MAPT P10636 4/20 0.37
USP2 O75604 2/20 0.37
ALOX12 P18054 2/20 0.37
GAA P10253 1/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
KCNA5 P22460 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HPGD P15428 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10149607 1.00 RECQL (0.39) RECQLALDH1A1MAPTUSP2ALOX12
SCHEMBL3143180 0.77 ALDH1A1 (0.35) RECQLALDH1A1MAPTUSP2GAA
SCHEMBL219983 0.77
SCHEMBL219982 0.77
SCHEMBL10149589 0.75 NPC1 (0.32) ALDH1A1MAPTUSP2NPC1MAPK1
SCHEMBL328593 0.74 RECQL (0.42) RECQLALDH1A1MAPTUSP2ALOX12
SCHEMBL454530 0.72
SCHEMBL454529 0.72
SCHEMBL9142690 0.72
SCHEMBL31531962 0.70 ALDH1A1 (0.46) RECQLALDH1A1MAPTUSP2ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0897914-B1 Process for the preparation of 2,5-disubstitued pyridines HOFFMANN LA ROCHE (CH) 2004-05-26 EP claimed
US-6080866-A A CHEMICAL INTERMEDIATES FOR ENDOTHELIN RECEPTOR ANTAGONISTS HOFFMANN-LA ROCHE INC. (US) 2000-06-27 US claimed
CN-1210105-A Process for preparation of 2,5-disubstituted pyridines HOFFMANN LA ROCHE (CH) 1999-03-10 CN claimed
EP-0897914-A1 Process for the preparation of 2,5-disubstitued pyridines F. HOFFMANN-LA ROCHE AG (CH) 1999-02-24 EP claimed
EP-0897914-B1 Process for the preparation of 2,5-disubstitued pyridines HOFFMANN LA ROCHE (CH) 2004-05-26 EP disclosed
CN-1103335-C Process for preparation of 2,5-disubstituted pyridines HOFFMANN LA ROCHE (CH) 2003-03-19 CN disclosed
US-6080866-A A CHEMICAL INTERMEDIATES FOR ENDOTHELIN RECEPTOR ANTAGONISTS HOFFMANN-LA ROCHE INC. (US) 2000-06-27 US disclosed
CN-1210105-A Process for preparation of 2,5-disubstituted pyridines HOFFMANN LA ROCHE (CH) 1999-03-10 CN disclosed
EP-0897914-A1 Process for the preparation of 2,5-disubstitued pyridines F. HOFFMANN-LA ROCHE AG (CH) 1999-02-24 EP disclosed
US-4547594-A REACTING AND ACYCLIC, OXO, NITRILE WITH METHYL LITHIUM, THEN HYDROLYSIS INTERNATIONAL FLAVORS & FRAGRANCES INC. (US) 1985-10-15 US disclosed
US-4517385-A FROM ALDEHYDE-NITRILE AND ACETONE, TOBACCO FLABOR INTERNATIONAL FLAVORS & FRAGRANCES INC. (US) 1985-05-14 US disclosed
US-4489009-A Process for producing solanone, norsolanadione and intermediates therefor INTERNATIONAL FLAVORS & FRAGRANCES INC. (US) 1984-12-18 US disclosed
US-4486588-A Cyclohexadiene carboxylate insecticide intermediates FMC CORPORATION (US) 1984-12-04 US disclosed
US-4483995-A ORGANOLEPTIC TOBACCO ADDITIVES INTERNATIONAL FLAVORS & FRAGRANCES INC. (US) 1984-11-20 US disclosed
US-4412083-A TOBACCO FLAVOR, ORGANOLEPTIC INTERNATIONAL FLAVORS & FRAGRANCES INC. (US) 1983-10-25 US disclosed