SCHEMBL6582309

SCHEMBL6582309

CC(C)C[C@H](NS(=O)(=O)Cc1ccccc1[N+](=O)[O-])C(=O)NC1CN(Cc2ccccc2)CC1=O

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSK P43235 15/20 0.44
CTSL P07711 10/20 0.44
CTSS P25774 6/20 0.44
SIGMAR1 Q99720 1/20 0.43
CTSB P07858 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6582315 0.87 CTSK (0.51) CTSKCTSLCTSSCTSB
SCHEMBL6578303 0.86 CTSK (0.65) CTSKCTSLCTSSCTSB
SCHEMBL6581006 0.85 SIGMAR1 (0.43) CTSKSIGMAR1
SCHEMBL6582321 0.80 CTSK (0.51) CTSKCTSLCTSSCTSB
SCHEMBL6582644 0.79 CTSK (0.45) CTSKCTSLCTSSCTSB
SCHEMBL6577997 0.77 CTSK (0.46) CTSKCTSLCTSSCTSB
SCHEMBL6580052 0.75 CTSK (0.69) CTSKCTSLCTSSCTSB
SCHEMBL6583959 0.73 CTSK (0.52) CTSKCTSLCTSSCTSB
SCHEMBL6580739 0.73 CTSK (0.56) CTSKCTSLCTSSCTSB
Lithium Ion SCHEMBL6582305 0.72 CTSK (0.53) CTSKCTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0936912-B1 INHIBITORS OF CYSTEINE PROTEASE SMITHKLINE BEECHAM CORP (US) 2004-02-11 EP claimed
EP-0936912-A4 INHIBITORS OF CYSTEINE PROTEASE SMITHKLINE BEECHAM CORP (US) 1999-10-13 EP disclosed
EP-0936912-A1 INHIBITORS OF CYSTEINE PROTEASE SMITHKLINE BEECHAM CORPORATION (US) 1999-08-25 EP disclosed
WO-1998005336-A1 INHIBITORS OF CYSTEINE PROTEASE SMITHKLINE BEECHAM CORPORATION (US) 1998-02-12 WO disclosed