SCHEMBL6582449

SCHEMBL6582449

Nc1ccc(S(=O)(=O)Nc2cc[nH]n2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.54
LMNA P02545 6/20 0.54
CYP2C19 P33261 3/20 0.54
KDM4E B2RXH2 2/20 0.53
NPSR1 Q6W5P4 2/20 0.53
ALDH1A1 P00352 4/20 0.51
MAPT P10636 3/20 0.51
ADRA1A P35348 1/20 0.51
HTR6 P50406 5/20 0.50
PDE4A P27815 1/20 0.50
AGO2 Q9UKV8 1/20 0.50
AURKA O14965 1/20 0.50
DHFR P00374 1/20 0.50
TSHR P16473 1/20 0.50
CYP3A4 P08684 3/20 0.49
CYP2C9 P11712 2/20 0.49
RAB9A P51151 1/20 0.49
KMT2A Q03164 1/20 0.49
APEX1 P27695 1/20 0.48
BLM P54132 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1093985 0.83 ALDH1A1 (0.50) LMNAKDM4EALDH1A1TSHRKMT2A
SCHEMBL11883949 0.81 POLB (0.55) SMN1; SMN2LMNAALDH1A1HTR6TSHR
SCHEMBL28113811 0.80 CA2 (0.53) SMN1; SMN2LMNAKDM4EALDH1A1MAPT
SCHEMBL5565365 0.78 CA12 (0.54) SMN1; SMN2LMNAALDH1A1MAPTCYP2C9
SCHEMBL11884662 0.78 HTR6 (0.52) SMN1; SMN2LMNACYP2C19KDM4ENPSR1
SCHEMBL28335271 0.75
SCHEMBL28176926 0.71 KMT2A (0.58) ALDH1A1KMT2ACA1CA2CA9
SCHEMBL11882075 0.71 L3MBTL1 (0.77) SMN1; SMN2LMNACYP2C19KDM4ENPSR1
SCHEMBL20503569 0.71 HTT (0.39) SMN1; SMN2LMNAKDM4EALDH1A1RAB9A
SCHEMBL11793140 0.70 CA1 (0.85) CYP2C19ALDH1A1MAPTHTR6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111763172-B Halosulfuron-methyl hapten and complete antigen as well as preparation method and application thereof 中国农业科学院农业质量标准与检测技术研究所 2022-04-08 CN disclosed
CN-111763172-A Halosulfuron-methyl hapten and complete antigen as well as preparation method and application thereof 中国农业科学院农业质量标准与检测技术研究所 2020-10-13 CN disclosed
EP-1257539-B1 AMINO PYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF OBESITY AND OTHER DISORDERS ORTHO MCNEIL PHARM INC (US) 2004-12-29 EP disclosed
US-6531478-B2 For therapy of eating disorder, obesity, bulimia nervosa, diabetes, binge eating, anorexia nervosa, dyslipidimia, hypertension, memory loss, epileptic seizures, migraine, sleep disturbances, pain, sexual/reproductive disorders KORDIK CHERYL P (US) 2003-03-11 US disclosed
EP-1257539-A2 AMINO PYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF OBESITY AND OTHER DISORDERS Ortho-Mcneil Pharmaceutical, Inc. (US) 2002-11-20 EP disclosed
US-20020065289-A1 Amino pyrazole derivatives useful for the treatment of obesity and other disorders KORDIK CHERYL P (US) 2002-05-30 US disclosed
WO-2001062737-A2 AMINO PYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF OBESITY AND OTHER DISORDERS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-08-30 WO disclosed
US-3769076-A ARYLSULONAMIDOPYRAZOLE AND IMIDAZOLE INTUMESCENT COATED ARTICLES CITIES SERVICE CO 1973-10-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020065289-A1 Amino pyrazole derivatives useful for the treatment of obesity and other disorders NPY5R, NPY1R, NPY4R SMN1; SMN2 4189/4885LMNA 3821/4885CYP2C19 279/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.