SCHEMBL6582799

SCHEMBL6582799

Cc1nccc(NCC2CCN(C(=O)CNc3cccc(C(=O)OC(C)(C)C)c3Cl)CC2)n1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.38
BRD4 O60885 1/20 0.37
PRMT5 O14744 1/20 0.37
TGFBR1 P36897 1/20 0.36
GRIN2B Q13224 8/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
SCD O00767 3/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
KDM4E B2RXH2 1/20 0.35
PKM P14618 1/20 0.35
PIM1 P11309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6583196 0.86 BRD4 (0.38) BRD4TGFBR1GRIN2BSCDKDM4E
SCHEMBL6586188 0.84 GRIN2B (0.41) GRIN2BCYP3A4CYP2D6CYP2C9SCD
SCHEMBL6582859 0.84 GRIN2B (0.46) BRD4GRIN2BCYP3A4CYP2D6CYP2C9
SCHEMBL6582400 0.84 SCD (0.41) BRD4TGFBR1GRIN2BSCDKDM4E
SCHEMBL6582862 0.83 SCD (0.43) CCNT1CDK9GRIN2BCYP3A4CYP2D6
SCHEMBL6584670 0.82 HTR1A (0.37)
SCHEMBL6581653 0.80 HTR1A (0.37)
SCHEMBL6582672 0.79 GRIN2B (0.39) GRIN2BCYP2D6CYP2C9SCD
SCHEMBL6580506 0.78 BCHE (0.34) TGFBR1GRIN2BSCD
SCHEMBL6582688 0.74 CYP2D6 (0.44) TGFBR1GRIN2BCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1455788-A1 1-GLYCINYL-4-AMINOMETHYL-PIPERIDINE DERIVATIVES AS FACTOR XA INHIBITORS ELI LILLY AND COMPANY (US) 2004-09-15 EP disclosed
WO-2003049737-A1 CHEMICAL COMPOUNDS ELI LILLY AND COMPANY (US) 2003-06-19 WO disclosed