SCHEMBL6582672

SCHEMBL6582672

CC(C)(C)OC(=O)c1cccc(NCC(=O)N2CCC(CCNc3ccncc3)CC2)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.39
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
SCD O00767 4/20 0.37
GPR119 Q8TDV5 9/20 0.37
CXCR3 P49682 1/20 0.36
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6582688 0.82 CYP2D6 (0.44) GRIN2BCYP2D6CYP2C9SCDADRA1A
SCHEMBL6583196 0.80 BRD4 (0.38) GRIN2BSCDGPR119ADRA1AADRA1B
SCHEMBL6580506 0.80 BCHE (0.34) GRIN2BSCDADRA1AADRA1B
SCHEMBL6582799 0.79 CCNT1 (0.38) GRIN2BCYP2D6CYP2C9SCD
SCHEMBL6581653 0.79 HTR1A (0.37)
SCHEMBL6582859 0.79 GRIN2B (0.46) GRIN2BCYP2D6CYP2C9SCDGPR119
SCHEMBL7096292 0.77 GRIN2B (0.52) GRIN2BCYP2D6CYP2C9
SCHEMBL6582400 0.76 SCD (0.41) GRIN2BSCDGPR119
SCHEMBL6584670 0.76 HTR1A (0.37)
SCHEMBL6535858 0.76 GPR119 (0.57) GRIN2BCYP2D6CYP2C9GPR119KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1455788-A1 1-GLYCINYL-4-AMINOMETHYL-PIPERIDINE DERIVATIVES AS FACTOR XA INHIBITORS ELI LILLY AND COMPANY (US) 2004-09-15 EP disclosed
WO-2003049737-A1 CHEMICAL COMPOUNDS ELI LILLY AND COMPANY (US) 2003-06-19 WO disclosed