SCHEMBL6583196

SCHEMBL6583196

CC(C)(C)OC(=O)c1cccc(NCC(=O)N2CCC(CNc3cccnn3)CC2)c1Cl

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.38
KDM4E B2RXH2 1/20 0.36
PKM P14618 1/20 0.36
GRIN2B Q13224 2/20 0.36
SCD O00767 6/20 0.36
GPR119 Q8TDV5 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
TGFBR1 P36897 1/20 0.35
FNTA P49354 2/20 0.35
FNTB P49356 2/20 0.35
PIM1 P11309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581653 0.89 HTR1A (0.37)
SCHEMBL6582799 0.86 CCNT1 (0.38) BRD4KDM4EPKMGRIN2BSCD
SCHEMBL6582859 0.82 GRIN2B (0.46) BRD4GRIN2BSCDGPR119PIM1
SCHEMBL5412796 0.81 SCD (0.45) GRIN2BSCD
SCHEMBL6582672 0.80 GRIN2B (0.39) GRIN2BSCDGPR119ADRA1AADRA1B
SCHEMBL6582400 0.80 SCD (0.41) BRD4KDM4EPKMGRIN2BSCD
SCHEMBL6584670 0.78 HTR1A (0.37)
SCHEMBL6582688 0.74 CYP2D6 (0.44) KDM4EPKMGRIN2BSCDADRA1A
SCHEMBL6580506 0.74 BCHE (0.34) GRIN2BSCDADRA1AADRA1BTGFBR1
SCHEMBL5410680 0.74 KDM4E (0.38) BRD4KDM4EPKMGRIN2BTGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1455788-A1 1-GLYCINYL-4-AMINOMETHYL-PIPERIDINE DERIVATIVES AS FACTOR XA INHIBITORS ELI LILLY AND COMPANY (US) 2004-09-15 EP disclosed
WO-2003049737-A1 CHEMICAL COMPOUNDS ELI LILLY AND COMPANY (US) 2003-06-19 WO disclosed