SCHEMBL6583301

SCHEMBL6583301

CCOc1cc(C2=NN(C(=O)c3cccc(NC(=O)c4cccc(NC(=O)c5ccc(Cl)cc5Cl)c4)c3)CCC2)ccc1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
LMNA P02545 2/20 0.49
PKM P14618 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
TP53 P04637 3/20 0.48
MAPT P10636 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
NFKB1 P19838 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47
PGR P06401 5/20 0.45
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
KMT2A Q03164 2/20 0.42
GRM5 P41594 1/20 0.41
MEN1 O00255 1/20 0.41
CES1 P23141 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6582145 0.96 TP53 (0.50) ALDH1A1LMNAPKMNPSR1TP53
SCHEMBL6585171 0.93 ALDH1A1 (0.55) ALDH1A1LMNAPKMNPSR1TP53
SCHEMBL6583372 0.92 ALDH1A1 (0.52) ALDH1A1LMNAPKMNPSR1MAPT
SCHEMBL6586320 0.90 ALDH1A1 (0.52) ALDH1A1LMNAPKMNPSR1TP53
SCHEMBL6583492 0.90 ALDH1A1 (0.51) ALDH1A1LMNAPKMNPSR1TP53
SCHEMBL6581858 0.89 SMN1; SMN2 (0.49) ALDH1A1LMNAPKMNPSR1TP53
SCHEMBL6584065 0.89 ALDH1A1 (0.51) ALDH1A1LMNAPKMNPSR1TP53
SCHEMBL6582371 0.89 NPC1 (0.49) ALDH1A1LMNAPKMNPSR1MAPT
SCHEMBL6585085 0.88 PGR (0.53) ALDH1A1LMNAPKMNPSR1TP53
SCHEMBL6585175 0.87 ALDH1A1 (0.51) ALDH1A1LMNAPKMNPSR1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194411-B1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2004-06-16 EP disclosed
US-6696446-B1 HETEROCYLCIC AMIDES SUCH AS N-(4-(3-(3-(3-ETHOXY-4-METHOXY PHENYL)-1,4,5,6-TETRAHYDRO-1-PYRIDAZINYLCARBONYL)PHENYLAMINO -CARBONYL)PHENYL)-4-NITROBENZAMIDE, SUED AS PHOSPHODIESTERASE INHIBITORSFOR PROPHYLAXIS OF ALLERGIES OR ASTHMA MERCK PATENT GMBH (DE) 2004-02-24 US disclosed
EP-1194411-A1 BENZOYLPYRIDAZINES MERCK PATENT GmbH (DE) 2002-04-10 EP disclosed
WO-2001004099-A1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2001-01-18 WO disclosed