SCHEMBL6583312

SCHEMBL6583312

O=C1CCCc2c(cccc2OCCCCl)N1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
DRD3 P35462 1/20 0.45
ADRB1 P08588 3/20 0.45
ADRB2 P07550 1/20 0.45
HTR1A P08908 1/20 0.45
OPRK1 P41145 1/20 0.45
MAPT P10636 2/20 0.43
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38
TRPM2 O94759 1/20 0.36
PARP1 P09874 1/20 0.36
LMNA P02545 2/20 0.36
TP53 P04637 1/20 0.36
KIF11 P52732 1/20 0.35
NPC1 O15118 1/20 0.35
MAPK13 O15264 1/20 0.35
MAPK12 P53778 1/20 0.35
MAPK11 Q15759 1/20 0.35
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9653164 0.92 ADRB1 (0.52) DRD2DRD4DRD3ADRB1ADRB2
SCHEMBL9653685 0.87 ADRB1 (0.51) DRD2DRD4DRD3ADRB1ADRB2
SCHEMBL9653135 0.86 ADRB1 (0.50) DRD2DRD4DRD3ADRB1ADRB2
SCHEMBL9389280 0.86 ADRB1 (0.52) DRD2DRD4DRD3ADRB1ADRB2
SCHEMBL6588799 0.84 DRD2 (0.61) DRD2DRD4DRD3ADRB1ADRB2
SCHEMBL18072426 0.79 ADRB2 (0.54) DRD2DRD4DRD3ADRB1ADRB2
SCHEMBL8054602 0.78 ALDH1A1 (0.46) DRD2DRD4DRD3ADRB1ADRB2
SCHEMBL9390026 0.78 DRD2 (0.61) DRD2DRD4DRD3ADRB1ADRB2
SCHEMBL885653 0.78 MAPT (0.49) ADRB1ADRB2HTR1AOPRK1MAPT
SCHEMBL30335516 0.78 ADRB1 (0.50) DRD2DRD4DRD3ADRB1ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0957100-B1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME KOWA CO (JP) 2004-10-27 EP disclosed
EP-0957100-A1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME Kowa Co., Ltd. (JP) 1999-11-17 EP disclosed