SCHEMBL6584231

SCHEMBL6584231

Cc1ccc(OCCCCCN2CCN(Cc3ccc4ccccc4n3)CC2)c2c1NC(=O)CC2

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.44
HTR1A P08908 9/20 0.44
HTR2A P28223 7/20 0.44
MAOA P21397 3/20 0.41
MAOB P27338 3/20 0.41
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6582756 0.99 DRD2 (0.45) DRD2HTR1AHTR2AMAOAMAOB
SCHEMBL6587330 0.97 DRD2 (0.43) DRD2HTR1AHTR2AMAOAMAOB
SCHEMBL6585890 0.97 DRD2 (0.43) DRD2HTR1AHTR2AMAOAMAOB
SCHEMBL6585521 0.96 HTR1A (0.42) DRD2HTR1AHTR2AMAOAMAOB
SCHEMBL6582486 0.94 DRD2 (0.41) DRD2HTR1AHTR2AMAOAMAOB
SCHEMBL6583995 0.94 MEN1 (0.46) DRD2HTR1AHTR2AMEN1MAPT
SCHEMBL6585920 0.91 MEN1 (0.43) DRD2HTR1AHTR2AMEN1MAPT
SCHEMBL7508996 0.85 DRD4 (0.40) DRD2HTR1AHTR2AMAOAMAOB
SCHEMBL6584859 0.84 HTR1A (0.41) DRD2HTR1AHTR2AMEN1MAPT
SCHEMBL6583201 0.84 DRD2 (0.41) DRD2HTR1AHTR2AMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0957100-B1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME KOWA CO (JP) 2004-10-27 EP disclosed
EP-0957100-A1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME Kowa Co., Ltd. (JP) 1999-11-17 EP disclosed