SCHEMBL6585920

SCHEMBL6585920

Cc1ccc(OCCN2CCCN(Cc3ccc4ccccc4n3)CC2)c2c1NC(=O)CC2

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43
HTR1A P08908 4/20 0.39
HTR7 P34969 1/20 0.39
HTR1D P28221 2/20 0.38
HTR1B P28222 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
FAAH O00519 1/20 0.38
DRD2 P14416 4/20 0.38
HTR2A P28223 1/20 0.37
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
MCHR1 Q99705 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6583995 0.97 MEN1 (0.46) MEN1MAPTKMT2AHTR1AHTR7
SCHEMBL6582486 0.96 DRD2 (0.41) MEN1MAPTKMT2AHTR1AHTR7
SCHEMBL6585890 0.95 DRD2 (0.43) HTR1ADRD2HTR2A
SCHEMBL6587330 0.94 DRD2 (0.43) HTR1ADRD2HTR2A
SCHEMBL6585521 0.93 HTR1A (0.42) MEN1MAPTKMT2AHTR1AHTR7
SCHEMBL6582756 0.92 DRD2 (0.45) MEN1MAPTKMT2AHTR1ADRD2
SCHEMBL6584231 0.91 DRD2 (0.44) MEN1MAPTKMT2AHTR1ADRD2
SCHEMBL7517500 0.85 HTR1A (0.44) MEN1MAPTKMT2AHTR1AHTR7
SCHEMBL6585099 0.85 GRM2 (0.45) MAPTDRD2
SCHEMBL6585787 0.84 MEN1 (0.43) MEN1MAPTKMT2AHTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0957100-B1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME KOWA CO (JP) 2004-10-27 EP disclosed
EP-0957100-A1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME Kowa Co., Ltd. (JP) 1999-11-17 EP disclosed