SCHEMBL6587589

SCHEMBL6587589

CCOc1cc(C2=NN(C(=O)c3ccc(NC(=O)c4ccc(NC(=O)c5ccccc5)cc4)cc3)CCC2)ccc1OC

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
POLB P06746 2/20 0.52
MAPT P10636 5/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
PGR P06401 5/20 0.48
LMNA P02545 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MCHR1 Q99705 2/20 0.47
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
MAOB P27338 1/20 0.44
TP53 P04637 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581435 0.96 KMT2A (0.49) ALDH1A1POLBMAPTMEN1KMT2A
SCHEMBL6581923 0.95 NPC1 (0.48) ALDH1A1POLBMAPTMEN1KMT2A
SCHEMBL6582201 0.93 GAA (0.51) ALDH1A1POLBMAPTPGRSMN1; SMN2
SCHEMBL6581784 0.93 ALDH1A1 (0.55) ALDH1A1POLBMAPTMEN1KMT2A
SCHEMBL6585136 0.93 ALDH1A1 (0.49) ALDH1A1POLBMAPTMEN1KMT2A
Benzoyl Chloride SCHEMBL7559384 0.93 NPC1 (0.48) ALDH1A1POLBMAPTMEN1KMT2A
SCHEMBL6601230 0.92 HTT (0.47) ALDH1A1POLBMAPTMEN1KMT2A
SCHEMBL6581226 0.92 PGR (0.54) ALDH1A1POLBMAPTPGRLMNA
SCHEMBL6584572 0.92 NPC1 (0.45) ALDH1A1POLBMAPTMEN1KMT2A
SCHEMBL6581583 0.92 ALDH1A1 (0.52) ALDH1A1POLBMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194411-B1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2004-06-16 EP disclosed
US-6696446-B1 HETEROCYLCIC AMIDES SUCH AS N-(4-(3-(3-(3-ETHOXY-4-METHOXY PHENYL)-1,4,5,6-TETRAHYDRO-1-PYRIDAZINYLCARBONYL)PHENYLAMINO -CARBONYL)PHENYL)-4-NITROBENZAMIDE, SUED AS PHOSPHODIESTERASE INHIBITORSFOR PROPHYLAXIS OF ALLERGIES OR ASTHMA MERCK PATENT GMBH (DE) 2004-02-24 US disclosed
EP-1194411-A1 BENZOYLPYRIDAZINES MERCK PATENT GmbH (DE) 2002-04-10 EP disclosed
WO-2001004099-A1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2001-01-18 WO disclosed