SCHEMBL6581232

SCHEMBL6581232

CCOc1cc(C2=NN(C(=O)c3ccc(NC(=O)c4cccc(N)c4)cc3)CCC2)ccc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.44
ALDH1A1 P00352 3/20 0.44
KMT2A Q03164 5/20 0.43
MAPT P10636 5/20 0.43
MEN1 O00255 3/20 0.43
TP53 P04637 1/20 0.42
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
GAA P10253 1/20 0.42
CASP1 P29466 1/20 0.42
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
HPSE Q9Y251 1/20 0.41
USP2 O75604 1/20 0.41
MAOB P27338 1/20 0.41
LMNA P02545 2/20 0.41
PKM P14618 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6583658 0.94 NPC1 (0.45) POLBALDH1A1KMT2AMAPTMEN1
SCHEMBL6584572 0.92 NPC1 (0.45) POLBALDH1A1KMT2AMAPTMEN1
SCHEMBL6587589 0.91 ALDH1A1 (0.52) POLBALDH1A1KMT2AMAPTMEN1
SCHEMBL6585136 0.91 ALDH1A1 (0.49) POLBALDH1A1KMT2AMAPTMEN1
SCHEMBL6581435 0.91 KMT2A (0.49) POLBALDH1A1KMT2AMAPTMEN1
SCHEMBL5202716 0.90 ALDH1A1 (0.49) POLBALDH1A1MAPTSMN1; SMN2GAA
SCHEMBL6581583 0.90 ALDH1A1 (0.52) POLBALDH1A1KMT2AMAPTMEN1
SCHEMBL6584628 0.89 PGR (0.47) POLBALDH1A1KMT2AMAPTMEN1
SCHEMBL6763155 0.89 ALDH1A1 (0.51) POLBALDH1A1KMT2AMAPTMEN1
SCHEMBL6767556 0.89 ALDH1A1 (0.47) POLBALDH1A1KMT2AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194411-B1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2004-06-16 EP disclosed
US-6696446-B1 HETEROCYLCIC AMIDES SUCH AS N-(4-(3-(3-(3-ETHOXY-4-METHOXY PHENYL)-1,4,5,6-TETRAHYDRO-1-PYRIDAZINYLCARBONYL)PHENYLAMINO -CARBONYL)PHENYL)-4-NITROBENZAMIDE, SUED AS PHOSPHODIESTERASE INHIBITORSFOR PROPHYLAXIS OF ALLERGIES OR ASTHMA MERCK PATENT GMBH (DE) 2004-02-24 US disclosed