SCHEMBL6584628

SCHEMBL6584628

CCOc1cc(C2=NN(C(=O)c3ccc(NC(=O)c4cccc(NC(=O)c5ccc(C)cc5)c4)cc3)CCC2)ccc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.47
NPC1 O15118 4/20 0.46
RAB9A P51151 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
ALDH1A1 P00352 3/20 0.46
GAA P10253 3/20 0.46
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.44
MAPT P10636 2/20 0.44
POLB P06746 2/20 0.43
TP53 P04637 1/20 0.43
CASP1 P29466 1/20 0.42
NPSR1 Q6W5P4 2/20 0.42
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CASP3 P42574 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581435 0.95 KMT2A (0.49) PGRNPC1RAB9ASMN1; SMN2NFKB1
SCHEMBL6583265 0.95 NPC1 (0.45) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6582201 0.94 GAA (0.51) PGRNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL6763155 0.94 ALDH1A1 (0.51) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6583333 0.94 KMT2A (0.49) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6581858 0.93 SMN1; SMN2 (0.49) PGRNPC1RAB9ASMN1; SMN2NFKB1
SCHEMBL6581923 0.93 NPC1 (0.48) PGRNPC1RAB9ASMN1; SMN2NFKB1
SCHEMBL6767556 0.92 ALDH1A1 (0.47) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
Benzoyl Chloride SCHEMBL7559384 0.92 NPC1 (0.48) PGRNPC1RAB9ASMN1; SMN2NFKB1
SCHEMBL6580950 0.92 NPC1 (0.45) NPC1RAB9ASMN1; SMN2NFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194411-B1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2004-06-16 EP disclosed
US-6696446-B1 HETEROCYLCIC AMIDES SUCH AS N-(4-(3-(3-(3-ETHOXY-4-METHOXY PHENYL)-1,4,5,6-TETRAHYDRO-1-PYRIDAZINYLCARBONYL)PHENYLAMINO -CARBONYL)PHENYL)-4-NITROBENZAMIDE, SUED AS PHOSPHODIESTERASE INHIBITORSFOR PROPHYLAXIS OF ALLERGIES OR ASTHMA MERCK PATENT GMBH (DE) 2004-02-24 US disclosed
EP-1194411-A1 BENZOYLPYRIDAZINES MERCK PATENT GmbH (DE) 2002-04-10 EP disclosed
WO-2001004099-A1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2001-01-18 WO disclosed