SCHEMBL6584810

SCHEMBL6584810

O=C1NC(c2ccncc2)=NC1(c1ccccc1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.54
BACE2 Q9Y5Z0 4/20 0.54
CYP2C9 P11712 3/20 0.54
BLM P54132 2/20 0.54
PMP22 Q01453 2/20 0.54
LMNA P02545 1/20 0.54
GLA P06280 1/20 0.54
THRB P10828 1/20 0.54
KMT2A Q03164 1/20 0.54
NOTUM Q6P988 1/20 0.42
MMP13 P45452 1/20 0.41
CTSD P07339 1/20 0.40
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
GSK3B P49841 2/20 0.36
CDC7 O00311 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6591928 0.89 BACE1 (0.61) BACE1BACE2CYP2C9BLMPMP22
SCHEMBL6588437 0.82 BACE1 (0.50) BACE1BACE2CYP2C9BLMPMP22
SCHEMBL6591279 0.81 BACE1 (0.53) BACE1BACE2CYP2C9BLMPMP22
SCHEMBL6589473 0.81 BACE1 (0.53) BACE1BACE2CYP2C9BLMPMP22
SCHEMBL6590512 0.81 BACE1 (0.49) BACE1BACE2CYP2C9BLMPMP22
SCHEMBL8235054 0.78 BACE1 (0.83) BACE1BACE2CYP2C9BLMPMP22
SCHEMBL6589904 0.78 BACE1 (0.53) BACE1BACE2CYP2C9BLMPMP22
SCHEMBL6599494 0.78 BACE1 (0.49) BACE1BACE2CYP2C9BLMPMP22
SCHEMBL6587050 0.77 LMNA (0.51) BACE1BACE2CYP2C9BLMPMP22
SCHEMBL6587379 0.76 BACE1 (0.47) BACE1BACE2CYP2C9BLMPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1066278-A4 IMIDAZOLONE ANORECTIC AGENTS: III. HETEROARYL DERIVATIVES BRISTOL MYERS SQUIBB CO (US) 2004-09-01 EP disclosed
EP-1066278-A1 IMIDAZOLONE ANORECTIC AGENTS: III. HETEROARYL DERIVATIVES Bristol-Myers Squibb Company (US) 2001-01-10 EP disclosed
WO-1999048887-A1 IMIDAZOLONE ANORECTIC AGENTS: III. HETEROARYL DERIVATIVES BRISTOL-MYERS SQUIBB COMPANY (US) 1999-09-30 WO disclosed